Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CDK12-IN-3 is a selective CDK12 inhibitor (IC50: 491 nM in an enzymatic assay).
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
25 mg | 約6-8 週間 | ¥ 349,000 |
50 mg | 約6-8 週間 | ¥ 454,500 |
100 mg | 約6-8 週間 | ¥ 574,000 |
説明 | CDK12-IN-3 is a selective CDK12 inhibitor (IC50: 491 nM in an enzymatic assay). |
ターゲット&IC50 | CDK12:491 nM |
In vitro | CDK12-IN-3 is a selective CDK12 inhibitor that is profiled across a panel of 352 kinases at 0.1 μM. CDK12-IN-3 shows potent inhibition of phosphorylation of Ser2 on the CTD repeat domain of RNA Pol II. It also shows growth inhibition of OV90 cells and acute cytotoxicity to THP1 cells. |
分子量 | 470.52 |
分子式 | C23H28F2N8O |
CAS No. | 2220184-50-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
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CDK12-IN-3 2220184-50-7 Cell Cycle/Checkpoint CDK CDK12IN3 CDK12 IN 3 CDK-12-IN-3 Inhibitor inhibitor inhibit