Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Chroman 1 is a potent inhibitor of ROCK1 (IC50 = 52 pM) and ROCK2 (IC50 = 1 pM).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 16,000 | |||
5 mg | 在庫あり | ¥ 39,500 | |||
10 mg | 在庫あり | ¥ 64,000 | |||
25 mg | 在庫あり | ¥ 117,500 | |||
50 mg | 在庫あり | ¥ 170,500 | |||
100 mg | 在庫あり | ¥ 226,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 44,500 |
説明 | Chroman 1 is a potent inhibitor of ROCK1 (IC50 = 52 pM) and ROCK2 (IC50 = 1 pM). |
ターゲット&IC50 | ROCK1:52 pM, ROCK2:1 pM, MRCK:150 nM |
In vitro | Chroman 1 also shows inhibitory activities against MRCK (IC50: 150 nM). However, it has no effect on PKA (IC50, > 20000 nM) or AKT1 (IC50, > 20000 nM). |
分子量 | 436.5 |
分子式 | C24H28N4O4 |
CAS No. | 1273579-40-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (114.55 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
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