Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Darbufelone (CI-1004) is a non-competitive dual inhibitor of PGF2α and LTB4. Dabfilon effectively inhibits PGHS-2 with a Ki of 10 μM and IC50s of 0.19 μM and 20 μM for PGHS-2 and PGHS-1.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
無料サンプル 1 mg | |||||
1 mg | 在庫あり | ¥ 14,500 | |||
5 mg | 在庫あり | ¥ 30,500 | |||
10 mg | 在庫あり | ¥ 51,500 | |||
25 mg | 在庫あり | ¥ 112,500 | |||
50 mg | 在庫あり | ¥ 164,000 | |||
100 mg | 在庫あり | ¥ 226,500 | |||
500 mg | 在庫あり | ¥ 454,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 43,500 |
説明 | Darbufelone (CI-1004) is a non-competitive dual inhibitor of PGF2α and LTB4. Dabfilon effectively inhibits PGHS-2 with a Ki of 10 μM and IC50s of 0.19 μM and 20 μM for PGHS-2 and PGHS-1. |
ターゲット&IC50 | PGHS-1:20 μM , PGHS-2:0.19 μM |
別名 | CI-1004 |
分子量 | 332.46 |
分子式 | C18H24N2O2S |
CAS No. | 139226-28-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45 mg/mL (135.35 mM)
You can also refer to dose conversion for different animals. 詳細
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Darbufelone 139226-28-1 GPCR/G Protein Immunology/Inflammation Prostaglandin Receptor LTR CI1004 CI-1004 CI 1004 Inhibitor inhibitor inhibit