Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
25 mg | 約8-10 週間 | ¥ 452,500 |
50 mg | 約8-10 週間 | ¥ 592,500 |
100 mg | 約8-10 週間 | ¥ 780,500 |
説明 | Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity. |
ターゲット&IC50 | D1 receptor:10 nM, D1 receptor:660 nM |
In vivo | Dihydrexidine shows poor oral bioavailability. It also has a relatively short half-life of 1 to 2 h [3]. Dihydrexidine hydrochloride (3 mg/kg; i.p.) yields dopamine D1 receptor agonist effects in vivo [4]. |
別名 | DAR-0100 |
分子量 | 267.32 |
分子式 | C17H17NO2 |
CAS No. | 123039-93-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
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Dihydrexidine 123039-93-0 GPCR/G Protein Neuroscience Dopamine Receptor DAR-0100 DAR0100 DAR 0100 Inhibitor inhibitor inhibit