Powder: -20°C for 3 years | In solvent: -80°C for 1 year
L 888607 Racemate is a selective antagonist of prostaglandin D2 receptor subtype 1 (DP1) (Kis: 132 nM and 17 nM for DP1 and thromboxane A2 receptor (TP), respectively).
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
25 mg | 約6-8 週間 | ¥ 248,000 |
50 mg | 約6-8 週間 | ¥ 323,500 |
100 mg | 約6-8 週間 | ¥ 457,000 |
説明 | L 888607 Racemate is a selective antagonist of prostaglandin D2 receptor subtype 1 (DP1) (Kis: 132 nM and 17 nM for DP1 and thromboxane A2 receptor (TP), respectively). |
ターゲット&IC50 | DP/DP1:132 nM (ki), TP:17 nM (ki) |
In vitro | L 888607 Racemate is actually 8-fold more effective on the TP receptor (Ki = 17 nM). L 888607 Racemate maintains a modest binding affinity for the DP1 receptor (Ki = 132 nM) . |
分子量 | 375.84 |
分子式 | C19H15ClFNO2S |
CAS No. | 1030017-51-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 6 mg/mL (15.96 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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L 888607 Racemate 1030017-51-6 Cell Cycle/Checkpoint Chromatin/Epigenetic Aurora Kinase Inhibitor inhibitor inhibit