Lisaftoclax is a dual Bcl-2 and Bcl-xl inhibitor (IC50: 2 nM and 5.9 nM) with antitumor activity.
| パッケージサイズ | 在庫状況 | 単価(税別) | |
|---|---|---|---|
| 1 mg | 在庫あり | ￥ 160000 | |
| 5 mg | 在庫あり | ￥ 305000 | |
| 10 mg | 在庫あり | ￥ 486000 | |
| 100 mg | 在庫あり | お問い合わせ | |
| 説明 | Lisaftoclax is a dual Bcl-2 and Bcl-xl inhibitor (IC50: 2 nM and 5.9 nM) with antitumor activity. |
| In vitro | Lisaftoclax shows IC50s of 5.5 nM and 6.4 nM in Bcl-2 dependent RS4 11 cells and Bcl-xl dependent Molm 13 cells[1]. |
| 別名 | APG-2575, Bcl-2/Bcl-xl inhibitor 1 |
| 分子量 | 882.42 |
| 分子式 | C45H48ClN7O8S |
| CAS No. | 2180923-05-9 |
Powder: -20°C for 3 years In solvent: -80°C for 2 years
DMSO: 225mg/mL (255mM), Need ultrasonic
( < 1 mg/ml refers to the product slightly soluble or insoluble )
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投与量変換You can also refer to dose conversion for different animals. 詳細
In vivo投与量計算 (透明溶液)計算器bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
