Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, antianxiety, antiemetic, hypotrophic, hypnotic and antihistamine effects, and can be used as a combination of norepinephrine and specific serotonin to treat depression.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 91,500 |
5 mg | 在庫あり | ¥ 223,000 |
10 mg | 在庫あり | ¥ 296,000 |
25 mg | 在庫あり | ¥ 447,500 |
50 mg | 在庫あり | ¥ 601,500 |
説明 | Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, antianxiety, antiemetic, hypotrophic, hypnotic and antihistamine effects, and can be used as a combination of norepinephrine and specific serotonin to treat depression. |
In vivo | The atypical antidepressant mianserin, administered at doses of 1, 5 and 10 mg/kg SC, dose-dependently increased up to about 6 times extracellular dopamine in the medial prefrontal cortex of the rat. Mianserin failed to modify extracellular dopamine in the nucleus accumbens. Mianserin also dose-dependently increased extracellular noradrenaline in the prefrontal cortex[1]. |
別名 | Lantanon, Lumin, Norval, Lerivon, Depnon |
分子量 | 264.36 |
分子式 | C18H20N2 |
CAS No. | 24219-97-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: Insoluble
DMSO: Soluble
You can also refer to dose conversion for different animals. 詳細
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Mianserin 24219-97-4 GPCR/G Protein Immunology/Inflammation Neuroscience Histamine Receptor Lantanon Lumin Norval Tolvon Lerivon Depnon Mianserine Inhibitor inhibitor inhibit