Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).
説明 | PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM). |
ターゲット&IC50 | D4 receptor:8.8 nM (ki) |
In vitro | PD 168568 dihydrochloride has good selective for D4 receptor(Ki of 1842 nM for D2 receptor)[1]. |
In vivo | PD 168568 dihydrochloride inhibit amphetamine stimulated locomotor activity in the rat[1]. |
別名 | PD 168568 (dihydrochloride) |
分子量 | 422.39 |
分子式 | C22H29Cl2N3O |
CAS No. | 1782532-06-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/mL (130.21 mM)
You can also refer to dose conversion for different animals. 詳細
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PD 168568 dihydrochloride 1782532-06-2 GPCR/G Protein Neuroscience Dopamine Receptor PD 168568 (dihydrochloride) PD 168568 PD168568 Dihydrochloride PD168568 PD-168568 PD-168568 Dihydrochloride PD 168568 Dihydrochloride Inhibitor inhibitor inhibit