Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PFI-2 is an effective, specific and cell-active lysine methyltransferase SETD7 inhibitor (Ki/IC50: 0.33/2 nM), 1000-fold selectivity over other methyltransferases and other non-epigenetic targets.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
5 mg | 約4-6 週間 | ¥ 19,000 |
10 mg | 約4-6 週間 | ¥ 30,000 |
25 mg | 約4-6 週間 | ¥ 58,500 |
50 mg | 約4-6 週間 | ¥ 103,000 |
100 mg | 約4-6 週間 | ¥ 185,500 |
説明 | PFI-2 is an effective, specific and cell-active lysine methyltransferase SETD7 inhibitor (Ki/IC50: 0.33/2 nM), 1000-fold selectivity over other methyltransferases and other non-epigenetic targets. |
ターゲット&IC50 | SETD7:2 nM |
別名 | PFI2, PFI 2, (R)-PFI-2 |
分子量 | 499.52 |
分子式 | C23H25F4N3O3S |
CAS No. | 1627676-59-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: 66 mg/mL (132.12 mM), Heating is recommended.
DMSO: >10 mM
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
PFI-2 1627676-59-8 Chromatin/Epigenetic Histone Methyltransferase PFI2 Inhibitor inhibit macrophage chronic kidney disease PFI 2 renal fibrosis inflammation (R)-PFI-2 SET domain containing lysine methyltransferase 7 (SETD7) inhibitor