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Alkaloids are a class of naturally occurring organic compounds that mostly contain basic nitrogen atoms, produced by a large variety of organisms including bacteria, fungi, plants, and animals. Alkaloids have a wide range of pharmacological activities including antimalarial (e.g. quinine), antiasthma (e.g. ephedrine), anticancer (e.g. homoharringtonine), cholinomimetic (e.g. galantamine), vasodilatory (e.g. vincamine), antiarrhythmic (e.g. quinidine), analgesic (e.g. morphine), antibacterial (e.g. chelerythrine), and antihyperglycemic activities (e.g. piperine). Many have found use in traditional or modern medicine, or as starting points for drug discovery. Other alkaloids possess psychotropic (e.g. psilocin) and stimulant activities (e.g. cocaine, caffeine, nicotine, theobromine), and have been used in entheogenic rituals or as recreational drugs. Alkaloids can be toxic too (e.g. atropine, tubocurarine).

カタログ番号 製品名
T3029 Sparteine sulfate Sparteine sulfate is a class 1a antiarrhythmic agent and a sodium channel blocker. It can chelate the bivalents calcium and magnesium.
T2S2104 Sinigrin hydrate 1. Sinigrin has antimicrobial activity. 2. Sinigrin exerts important anti-proliferative activities in carcinogen-induced hepatocarcinogenesis in rats, and highli...
TN1012 Febrifugine Febrifugine is an effective coccidiostat, possesses schizonticide props; it and its derivatives shows high degree of antimalarial activity but use limited by tox...
T4110 Perivine Perivine may resolve the instability of the retinoblastoma-associated proteins (RbAp48) complex and thus be used in Alzheimer's disease therapy. Perivine, vobasi...
T4912 Jatrorrhizine chloride Jatrorrhizine chloride is a potent and orally active uptake-2 transporter inhibitor. It exhibits a critical neuroprotective role in H2O2-induced apoptosis via in...
T4S0083 Protostemonine 1. Protostemonine has anti-inflammatory activity, it effectively attenuates LPS-induced inflammatory responses in vitro and in vivo; the beneficial effects are a...
TJS1226 Aristolactam I A natural compound from the herbs of Aristolochia debilis Sieb. et Zucc
T36115 Colchicoside Colchicoside is extracted from Gloriosa superba and shows efficacy in a murine model of pancreatic adenocarcinoma.
T8304 Anisodamine Hydrobromide Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
T8306 Epiberberine chloride Epiberberine chloride is an alkaloid isolated from Coptis chinensis, acts as a potent AChE and BChE inhibitor, and a non-competitive BACE1 inhibitor (IC50s: 1.07...
T4183 Lavendustin A lavendustin A is a potent, cell-permeable inhibitor of epidermal growth factor receptor (EGFR) tyrosine kinase.
TN7211 Tetrahydroharmine Tetrahydroharmine is a natural product found in the stems and large branches of Banisteriopsis caapi cultivar Da Vine. Tetrahydroharmine is a Monoamine oxidase A...
T2173 Veratridine Veratridine is a benzoate-cevane found in Veratrum and Schoenocaulon. It activates sodium channels to stay open longer than normal.
T1607 Hydrastinine hydrochloride Hydrastinine hydrochloride is a semisynthetic alkaloid from the hydrolysis of the alkaloid Hydrastine, used as a haemostatic drug.
T2S0058 6-Ethoxychelerythrine 6-Ethoxychelerythrine has anti-bacterial activity, it exhibited strong activity against Aspergillus fumigatus and methicillin-resistant Staphylococcus aureus (MR...
T2782 Catharanthine Catharanthine suppresses nicotinic receptor-mediated diaphragm contractions (IC50=59.6 μM).
T3S0804 Worenine Worenine is used in the a flurophore switched probe which aids in correction of an abasic site (AP site) caused by the removal of a damaged base in DNA.
TCS2336 Evodine 1. Evodine has antinociceptive activity.
TN2549 1-Methoxycarbonyl-β-carboline 1-Methoxycarbonyl-β-carboline is an alkaloid from Ailanthus altissima.
TN2460 12-Ethyl-9-hydroxycamptothecin 7-Ethyl-10-Hydroxy-Camptothecin is a natural product isolated from Camptotheca acuminata Decne
TCS2185 Yohimbine Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
T3022 Anhydrovinblastine 3', 4'-Anhydrovinblastine is an antineoplastic agent.
TN6787 N-noratherosperminine N-noratherosperminine is a alkaloid extract of the stem bark of Cryptocarya nigra.
TN1139 Dehydrocavidine Dehydrocavidine has antitumor activity, it inhibits MCF-7 cell proliferation by inducing apoptosis mediated by regulating Bax/Bcl-2, activating caspases as well ...
T3S0626 Denudatine 1. Denudatine has effects on action potential of ventricular fibers and has inhibition on arrhythmogenic action of aconitine.
TJS2216 Aurantiamide acetate Aurantiamide acetate was isolated from the fermentation broth of Aspergillus penicilloides for the first time. Aurantiamide acetate is a selective and orally act...
T3023 Catharanthine sulfate Catharanthine inhibits nicotinic receptor-mediated diaphragm contractions.
T67708 Thiolutin Thiolutin is an inhibitor of endothelial cell adhesion and produced by Streptomyces. Thiolutin shows antibiotic and anti-angiogenic properties. Thiolutin induces...
PDK0060 Pseudotropine Pseudotropine can cause hepatic necrosis and gastritis with ulceration or erosions.
PDK0014 3-Methylxanthine 3-Methylxanthine, a xanthine derivative, is a cyclic guanosine monophosphate (GMP) inhibitor, with an IC50 of 920 μM on guinea-pig isolated trachealis muscle.3-M...
TN1012L Febrifugine dihydrochloride Febrifugine dihydrochloride is a biochemical with therapeutic activity regarding malaria, cancer, fibrosis and inflammatory diseases.
TJS0123 Guvacine ethyl ester Arecoline is found in nuts. Arecoline is isolated from betel nuts Arecoline is an alkaloid natural product found in the areca nut, the fruit of the areca palm (A...
TN2027 Oxysanguinarine Oxysanguinarine possesses antiplatelet aggregation activity, it has potential inhibitory properties against dengue virus.
TN2298 Vincosamide Vincosamide is an alkaloid from Psychotria leiocarpa extract, inhibits the acetylcholinesterase (AChE) activity with anti-inflammatory activity. Vincosamide can ...
T5784 Topotecan Topotecan is a Topoisomerase I inhibitor,and is an antineoplastic agent used to treat ovarian cancer that works by inhibiting DNA topoisomerases.
TN2285 DL-Tryptophan Tryptophan containing dipeptides are interesting ingredients for functional foods as a natural prevention for hypertension with reduced side effects due to its s...
TC0014 Trachelanthine Trachelanthine is a natural product from Eupatorium fortunei.
TN3695 Coniine hydrochloride Coniine hydrochloride, a polyketide-derived alkaloid, is poisonous to humans and animals. It is a nicotinic acetylcholine receptor antagonist, which leads to inh...
TN2213 Imperialine 3-β-D-glucoside Imperialine 3-β-D-glucoside is a natural product. Imperialine 3-β-D-glucoside may exhibit anti-tumor properties against multi-drug resistant tumor cells.
Fr13711 Tropinone Tropinone used as an intermediate in the synthesis of atropine sulfate, and is a decane alkaloid.
Fr16605 Lupinine Lupinine is an alkaloid capable of counteracting ethanol anesthesia. Lupinine is an AChE and BChE inhibitor and potential CD69 activator found in species of Lora...
TN1754 Hypaconine Hypaconine is a C19-diterpenoid alkaloid isolated from Aconitum and Delphinium spp. It exhibits strong cardiac activity.
TN1474 Caulilexin C Caulilexin C shows inhibitory activity on human Acyl CoA: cholesterol transferase I (hACATI) and on human Acyl CoA: cholesterol transferase 2 (hACAT2) at 100 mug...
TC0022 Desoxypeganine Desoxypeganine is an inhibitor of cholinesterase. It acting preferentially on butyrylcholinesterase, and as a selective inhibitor of monoamine oxidase A but not ...
TN1353 N-Benzyllinoleamide N-Benzyllinoleamide is a natural product isolated from Lepidium meyenii Walp, has pharmaceutical property against exercise-induced fatigue.
Fr16741 Oxindole Oxindole is an aromatic heterocyclic building block. 2-indolinone derivatives have become lead compounds in the research of kinase inhibitors.Oxindole structure ...
TC0039 Vasicinone Vasicinone may act as a hepatoprotective agent. (±)-Vasicinone has significant antitussive, expectorant, and bronchodilating activities, which can be used to tre...
T5810 TABERSONINE HYDROCHLORIDE TABERSONINE HYDROCHLORIDE is a natural product extracted from the bean of Voacanga africana, is a potent inhibitor against Aβ(1 42) aggregation and toxicity.
T0130 Physostigmine Salicylate Physostigmine, a parasympathomimetic alkaloid, is a reversible cholinesterase inhibitor. It extracts from the Calabar bean.
T3002 Piperine Piperine (1-Piperoylpiperidine), a alkaloid, has been used in trials studying the treatment of multiple myeloma and deglutition disorders.
Sparteine sulfate
T3029
Sparteine sulfate is a class 1a antiarrhythmic agent and a sodium channel blocker. It can chelate the bivalents calcium and magnesium.
Sinigrin hydrate
T2S2104
1. Sinigrin has antimicrobial activity. 2. Sinigrin exerts important anti-proliferative activities in carcinogen-induced hepatocarcinogenesis in rats, and highli...
Febrifugine
TN1012
Febrifugine is an effective coccidiostat, possesses schizonticide props; it and its derivatives shows high degree of antimalarial activity but use limited by tox...
Perivine
T4110
Perivine may resolve the instability of the retinoblastoma-associated proteins (RbAp48) complex and thus be used in Alzheimer's disease therapy. Perivine, vobasi...
Jatrorrhizine chloride
T4912
Jatrorrhizine chloride is a potent and orally active uptake-2 transporter inhibitor. It exhibits a critical neuroprotective role in H2O2-induced apoptosis via in...
Protostemonine
T4S0083
1. Protostemonine has anti-inflammatory activity, it effectively attenuates LPS-induced inflammatory responses in vitro and in vivo; the beneficial effects are a...
Aristolactam I
TJS1226
A natural compound from the herbs of Aristolochia debilis Sieb. et Zucc
Colchicoside
T36115
Colchicoside is extracted from Gloriosa superba and shows efficacy in a murine model of pancreatic adenocarcinoma.
Anisodamine Hydrobromide
T8304
Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
Epiberberine chloride
T8306
Epiberberine chloride is an alkaloid isolated from Coptis chinensis, acts as a potent AChE and BChE inhibitor, and a non-competitive BACE1 inhibitor (IC50s: 1.07...
lavendustin A
T4183
lavendustin A is a potent, cell-permeable inhibitor of epidermal growth factor receptor (EGFR) tyrosine kinase.
Tetrahydroharmine
TN7211
Tetrahydroharmine is a natural product found in the stems and large branches of Banisteriopsis caapi cultivar Da Vine. Tetrahydroharmine is a Monoamine oxidase A...
Veratridine
T2173
Veratridine is a benzoate-cevane found in Veratrum and Schoenocaulon. It activates sodium channels to stay open longer than normal.
Hydrastinine hydrochloride
T1607
Hydrastinine hydrochloride is a semisynthetic alkaloid from the hydrolysis of the alkaloid Hydrastine, used as a haemostatic drug.
6-Ethoxychelerythrine
T2S0058
6-Ethoxychelerythrine has anti-bacterial activity, it exhibited strong activity against Aspergillus fumigatus and methicillin-resistant Staphylococcus aureus (MR...
Catharanthine
T2782
Catharanthine suppresses nicotinic receptor-mediated diaphragm contractions (IC50=59.6 μM).
Worenine
T3S0804
Worenine is used in the a flurophore switched probe which aids in correction of an abasic site (AP site) caused by the removal of a damaged base in DNA.
Evodine
TCS2336
1. Evodine has antinociceptive activity.
1-Methoxycarbonyl-β-carboline
TN2549
1-Methoxycarbonyl-β-carboline is an alkaloid from Ailanthus altissima.
12-Ethyl-9-hydroxycamptothecin
TN2460
7-Ethyl-10-Hydroxy-Camptothecin is a natural product isolated from Camptotheca acuminata Decne
Yohimbine
TCS2185
Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
Anhydrovinblastine
T3022
3', 4'-Anhydrovinblastine is an antineoplastic agent.
N-noratherosperminine
TN6787
N-noratherosperminine is a alkaloid extract of the stem bark of Cryptocarya nigra.
Dehydrocavidine
TN1139
Dehydrocavidine has antitumor activity, it inhibits MCF-7 cell proliferation by inducing apoptosis mediated by regulating Bax/Bcl-2, activating caspases as well ...
Denudatine
T3S0626
1. Denudatine has effects on action potential of ventricular fibers and has inhibition on arrhythmogenic action of aconitine.
Aurantiamide acetate
TJS2216
Aurantiamide acetate was isolated from the fermentation broth of Aspergillus penicilloides for the first time. Aurantiamide acetate is a selective and orally act...
Catharanthine sulfate
T3023
Catharanthine inhibits nicotinic receptor-mediated diaphragm contractions.
Thiolutin
T67708
Thiolutin is an inhibitor of endothelial cell adhesion and produced by Streptomyces. Thiolutin shows antibiotic and anti-angiogenic properties. Thiolutin induces...
Pseudotropine
PDK0060
Pseudotropine can cause hepatic necrosis and gastritis with ulceration or erosions.
3-Methylxanthine
PDK0014
3-Methylxanthine, a xanthine derivative, is a cyclic guanosine monophosphate (GMP) inhibitor, with an IC50 of 920 μM on guinea-pig isolated trachealis muscle.3-...
Febrifugine dihydrochloride
TN1012L
Febrifugine dihydrochloride is a biochemical with therapeutic activity regarding malaria, cancer, fibrosis and inflammatory diseases.
Guvacine ethyl ester
TJS0123
Arecoline is found in nuts. Arecoline is isolated from betel nuts Arecoline is an alkaloid natural product found in the areca nut, the fruit of the areca palm (A...
Oxysanguinarine
TN2027
Oxysanguinarine possesses antiplatelet aggregation activity, it has potential inhibitory properties against dengue virus.
Vincosamide
TN2298
Vincosamide is an alkaloid from Psychotria leiocarpa extract, inhibits the acetylcholinesterase (AChE) activity with anti-inflammatory activity. Vincosamide can ...
Topotecan
T5784
Topotecan is a Topoisomerase I inhibitor,and is an antineoplastic agent used to treat ovarian cancer that works by inhibiting DNA topoisomerases.
DL-Tryptophan
TN2285
Tryptophan containing dipeptides are interesting ingredients for functional foods as a natural prevention for hypertension with reduced side effects due to its s...
Trachelanthine
TC0014
Trachelanthine is a natural product from Eupatorium fortunei.
Coniine hydrochloride
TN3695
Coniine hydrochloride, a polyketide-derived alkaloid, is poisonous to humans and animals. It is a nicotinic acetylcholine receptor antagonist, which leads to inh...
Imperialine 3-β-D-glucoside
TN2213
Imperialine 3-β-D-glucoside is a natural product. Imperialine 3-β-D-glucoside may exhibit anti-tumor properties against multi-drug resistant tumor cells.
Tropinone
Fr13711
Tropinone used as an intermediate in the synthesis of atropine sulfate, and is a decane alkaloid.
Lupinine
Fr16605
Lupinine is an alkaloid capable of counteracting ethanol anesthesia. Lupinine is an AChE and BChE inhibitor and potential CD69 activator found in species of Lora...
Hypaconine
TN1754
Hypaconine is a C19-diterpenoid alkaloid isolated from Aconitum and Delphinium spp. It exhibits strong cardiac activity.
Caulilexin C
TN1474
Caulilexin C shows inhibitory activity on human Acyl CoA: cholesterol transferase I (hACATI) and on human Acyl CoA: cholesterol transferase 2 (hACAT2) at 100 mug...
Desoxypeganine
TC0022
Desoxypeganine is an inhibitor of cholinesterase. It acting preferentially on butyrylcholinesterase, and as a selective inhibitor of monoamine oxidase A but not ...
N-Benzyllinoleamide
TN1353
N-Benzyllinoleamide is a natural product isolated from Lepidium meyenii Walp, has pharmaceutical property against exercise-induced fatigue.
Oxindole
Fr16741
Oxindole is an aromatic heterocyclic building block. 2-indolinone derivatives have become lead compounds in the research of kinase inhibitors.Oxindole structure ...
Vasicinone
TC0039
Vasicinone may act as a hepatoprotective agent. (±)-Vasicinone has significant antitussive, expectorant, and bronchodilating activities, which can be used to tr...
TABERSONINE HYDROCHLORIDE
T5810
TABERSONINE HYDROCHLORIDE is a natural product extracted from the bean of Voacanga africana, is a potent inhibitor against Aβ(1 42) aggregation and toxicity.
Physostigmine Salicylate
T0130
Physostigmine, a parasympathomimetic alkaloid, is a reversible cholinesterase inhibitor. It extracts from the Calabar bean.
Piperine
T3002
Piperine (1-Piperoylpiperidine), a alkaloid, has been used in trials studying the treatment of multiple myeloma and deglutition disorders.
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