| T9833 |
Opiranserin hydrochloride
|
1440796-75-7
|
98%
|
|
|
Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM, ...
|
| T36949 |
Niaprazine
|
27367-90-4
|
98%
|
|
|
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for s...
|
| T22313 |
Dolasetron Mesylate
|
115956-13-3
|
98%
|
|
|
Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea following chemothera...
|
| T21011 |
Buspirone
|
36505-84-7
|
98%
|
|
|
Buspirone (Buspirone free base) is an azaspiro compound which has a role as an anxiolytic drug, a sedative, a serotonergic agonist and an EC 3.4.21.26 (prolyl ol...
|
| T22904 |
L-745870 trihydrochloride
|
866021-03-6
|
98%
|
|
|
L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.
|
| T4118 |
SB 271046 hydrochloride
|
209481-24-3
|
98%
|
|
|
SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist (pKi values are 9.02-8.92, 6.35, 6.55, 6.27 at 5-HT6, 5-HT1A, 5-HT1D and D3, an...
|
| T37197 |
5-HT1A modulator 2 hydrochloride
|
3880-76-0
|
98%
|
|
|
5-HT1A modulator 2 hydrochloride, a derivative of 8-OH-DPAT , is a modulator of 5-HT1A with a Ki of 53 nM for 5-HT1A binding[1].
[1]. Naiman, N.,et al. 2-(Alkyla...
|
| T28531 |
Facinicline hydrochloride
|
677305-02-1
|
98%
|
|
|
Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = 6 nM) and an antagonist of 5-HT3(Ki = 1.2 nM). ...
|
| T1066L |
Ketanserin tartrate
|
83846-83-7
|
98%
|
|
|
Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist with antihypertensive activity, inhibits serotonin-induced vaso...
|
| T22689 |
CP94253 hydrochloride
|
845861-39-4
|
98%
|
|
|
CP94253 hydrochloride (CP 94253 hydrochloride) is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, a...
|
| T12847 |
SB-616234-A
|
908601-49-0
|
98%
|
|
|
SB-616234A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant activity.
|
| TN1470 |
Cassiaside B2
|
218155-40-9
|
98%
|
|
|
Cassiaside B2 is an inhibitor of protein tyrosine phosphatase 1B (PTP1B) and human monoamine oxidase A (hMAO-A).Cassiaside B2 is an agonist of the 5-HT2C recepto...
|
| T1156 |
Palonosetron hydrochloride
|
135729-62-3
|
98%
|
|
|
Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.
|
| T2092 |
Amitifadine hydrochloride
|
410074-74-7
|
98%
|
|
|
Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
|
| T8385 |
Metoclopramide hydrochloride hydrate
|
54143-57-6
|
98%
|
|
|
Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction. It...
|
| T0338 |
Minaprine
|
25905-77-5
|
98%
|
|
|
Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.
|
| T22671 |
CJ 033466
|
519148-48-2
|
98%
|
|
|
CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.
|
| T23396 |
ST1936
|
1210-81-7
|
98%
|
|
|
ST1936 (ST 1936 oxalate) is a selective and potent 5-HT6 receptor agonist that inhibits human 5-HT6, 5-HT7, and 5-HT2B receptors, and stimulates cAMP, Ca2+, ERK1...
|
| T15270 |
Fananserin
|
127625-29-0
|
98%
|
|
|
Fananserin is an effective, selective and oral active antagonist of 5-HT2 (Ki = 0.37 nM for the rat 5-HT2A). Fananserin is an antagonist of human D4 receptor (Ki...
|
| T0113 |
Mebhydrolin napadisylate
|
6153-33-9
|
|
|
|
Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic derm...
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