T7320 |
Tozadenant
|
870070-55-6
|
98%
|
|
Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)
|
T0070 |
Pentoxifylline
|
6493-05-6
|
98%
|
|
Pentoxifylline (PTX) modulates immunologic activity by stimulating cytokine production. Pentoxifylline is a methylxanthine derivative that inhibits phosphodieste...
|
T4668 |
ABT-702 dihydrochloride
|
1188890-28-9
|
98%
|
|
ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.
|
T21017 |
5'-Amino-5'-deoxyadenosine
|
14365-44-7
|
98%
|
|
5'-Amino-5'-deoxyadenosine (NH2dAdo) is an adenosine kinase inhibitor targeting malignant tumors of the inert lymphatic system with antitumor and anticancer effe...
|
T4290 |
Preladenant
|
377727-87-2
|
98%
|
|
Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine ...
|
T15418 |
GS-6201
|
752222-83-6
|
98%
|
|
GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors with a ...
|
T0480 |
Doxofylline
|
69975-86-6
|
98%
|
|
Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofy...
|
T21620 |
Adenosine receptor antagonist 4
|
133240-06-9
|
98%
|
|
Adenosine receptor antagonist 4 is an adenosine receptor antagonist.
|
T12107 |
MRS-3777 hemioxalate
|
1186195-57-2
|
98%
|
|
MRS-3777 hemioxalate is a selective adenosine A3 receptor antagonist that reverses the anti-injury perception effects of its corresponding agonist and can be use...
|
T14078 |
AB928
|
2239273-34-6
|
98%
|
|
AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
|
T7188 |
Piclidenoson
|
152918-18-8
|
98%
|
|
Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.
|
T27076 |
8-Cyclopentyl-1,3-dimethylxanthine
|
35873-49-5
|
98%
|
|
8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.
|
T22489 |
2'-MeCCPA
|
205171-12-6
|
98%
|
|
2'-MeCCPA is a potent and highly selective A1 adenosine receptor (A1AR) agonist with a K-value of 1.8 nM for AR.2'-MeCCPA inhibits trichostatin-stimulated adenyl...
|
T34914 |
Trabodenoson
|
871108-05-3
|
98%
|
|
Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.
|
T15715 |
LAS101057
|
925676-48-8
|
98%
|
|
LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.
|
T29112 |
VPC171
|
1018830-99-3
|
98%
|
|
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
|
T16263 |
N6-Cyclopentyladenosine
|
41552-82-3
|
98%
|
|
N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of ...
|
T8613 |
1-Ethyl-6-aminouracil
|
41862-09-3
|
|
|
1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high affi...
|
T72067 |
DPTN dihydrochloride
|
325767-87-1
|
100%
|
|
DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.
|
T10248 |
Adenosine antagonist-1
|
431040-19-6
|
100%
|
|
Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.
|