T16759 |
Ritanserin
|
87051-43-2
|
98%
|
|
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine ...
|
T22905 |
L748337
|
244192-94-7
|
98%
|
|
L748337 is a competitive and potent β3-adrenoceptor antagonist that inhibits the action of β3-, β2-, and β1-adrenoceptors, activates MAPK signaling, promotes pho...
|
T36949 |
Niaprazine
|
27367-90-4
|
98%
|
|
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for s...
|
T5954 |
Methyldopa hydrate
|
41372-08-1
|
98%
|
|
Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension. It inhibits the sym...
|
T7164 |
Levalbuterol tartrate
|
661464-94-4
|
98%
|
|
Levalbuterol tartrate (Levosalbutamol tartrate) is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
|
T0226 |
Betaxolol hydrochloride
|
63659-19-8
|
98%
|
|
Betaxolol hydrochloride (SL 75212 HCl) is a cardioselective beta-blocker used in the treatment of hypertension.Betaxolol hydrochloride has not been linked to ins...
|
T12444 |
Phentolamine Analogue 1
|
47142-51-8
|
98%
|
|
Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.
|
T6519 |
Gramine
|
87-52-5
|
98%
|
|
Gramine (Donaxine), a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4...
|
T23382 |
Spiroxatrine
|
1054-88-2
|
98%
|
|
Spiroxatrine (R 5188) is a selective and potent 5-HT1α and α2-adrenergic dual antagonist with sedative activity and inhibitory effects on 5-HT1α, 5-HT1 β, 5-HT2,...
|
T24579 |
Oxyfedrine L-form HCl
|
16777-42-7
|
98%
|
|
Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.
|
T6860 |
ICI-118551 Hydrochloride
|
1217094-53-5
|
98%
|
|
ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors...
|
T0365 |
Thioridazine hydrochloride
|
130-61-0
|
98%
|
|
Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4 selecti...
|
T0185 |
Escitalopram
|
128196-01-0
|
98%
|
|
Escitalopram (Seroplex) is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing e...
|
T0248 |
Clorprenaline hydrochloride
|
6933-90-0
|
98%
|
|
Clorprenaline hydrochloride (Clorprenaline HCl) is a beta-2 adrenergic agonist with bronchodilator activity.
|
T21447 |
Tolazoline
|
59-98-3
|
98%
|
|
Tolazoline (Benzalolin), a non-selective competitive α-adrenergic receptor antagonist, is used as a vasodilator to treat spasms of peripheral blood vessels. It h...
|
T2547 |
Droxidopa
|
23651-95-8
|
98%
|
|
Droxidopa (L-DOPS) is an orally available prodrug of norepinephrine that is used in the treatment of symptomatic orthostatic hypotension due to neurogenic causes...
|
T10631 |
Bucindolol
|
71119-11-4
|
98%
|
|
Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.
|
T22904 |
L-745870 trihydrochloride
|
866021-03-6
|
98%
|
|
L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.
|
T5471 |
GUANABENZ
|
5051-62-7
|
98%
|
|
GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.
|
T10998 |
Deriglidole
|
122830-14-2
|
98%
|
|
Deriglidole (SL 86-0715) is a peripheral adrenergic receptor antagonist that is a selective inhibitor of alpha2 receptors. Deriglidole inhibits colistin and Idaz...
|