| T8592 |
CTK8A3536
|
926228-58-2
|
98%
|
|
|
CTK8A3536 ((2-MORPHOLIN-4-YL-4-PHENYL-1,3-THIAZOL-5-YL)METHANOL) is an inhibitor of Androgen receptor.
|
| T19450 |
N-desmethyl Enzalutamide
|
1242137-16-1
|
98%
|
|
|
N-desmethyl Enzalutamide (N-desmethyl MDV 3100) is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide. N-desmethyl Enzalutamide demon...
|
| T19470 |
Nandrolone propionate
|
7207-92-3
|
98%
|
|
|
Nandrolone propionate is an anabolic steroid action primarily consisting of androgenic and nitrogen-retentive properties.
|
| T6829 |
EPI-001
|
227947-06-0
|
98%
|
|
|
EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ～6 μM and a selective PPAR-gamma modulator.
|
| T20625 |
Prochloraz
|
67747-09-5
|
98%
|
|
|
Prochloraz (Prelude) is a broad-spectrum contact imidazole fungicide. Prochloraz inhibits human placental microsomal aromatase in vitro (IC50 = 40 nM). Prochlora...
|
| T2408 |
Ostarine
|
841205-47-8
|
98%
|
|
|
Ostarine (MK-2866) is a non-steroidal agent with anabolic activity. Selective androgen receptor modulator (SARM) GTx-024 is designed to work like testosterone, t...
|
| T28502 |
Ralaniten
|
1203490-23-6
|
98%
|
|
|
Ralaniten (EPI-002) is a potent, specific, and orally active antagonist of the androgen receptor N-terminal structural domain (AR-NTD).Ralaniten inhibits AR tran...
|
| T6915 |
Darolutamide
|
1297538-32-9
|
98%
|
|
|
Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).
|
| T7690 |
2-hydroxy Flutamide
|
52806-53-8
|
98%
|
|
|
2-hydroxy Flutamide is competitive inhibition of androgen receptor (AR) for the treatment of prostate cancer
|
| TN1067 |
Galloylpaeoniflorin
|
122965-41-7
|
98%
|
|
|
Galloylpaeoniflorin (6'-O-Galloyl paeoniflorin) may be developed as a cytoprotector against ROS-mediated oxidative stress. Galloylpaeoniflorin is also an inhibti...
|
| T39695 |
ARD-2128
|
2222111-87-5
|
98%
|
|
|
ARD-2128 is a highly potent, orally bioavailable PROTAC (proteolysis-targeting chimera) degrader of the androgen receptor (AR), effectively diminishing AR protei...
|
| T8860 |
DSRM-3716
|
58142-99-7
|
98%
|
|
|
Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery of a...
|
| T24943 |
VPC-14228
|
19983-28-9
|
98%
|
|
|
VPC-14228 is a specific AR-DBD inhibitor that acts by inhibiting both Y594A and Q592A mutants.
|
| T16090 |
MK-0773
|
606101-58-0
|
98%
|
|
|
MK-0773 (PF-05314882) is a selective androgen receptor modulator that binds to AR (IC50: 6.6 nM) for the study of diseases caused by endocrine abnormalities.
|
| T10359 |
AR antagonist 1
|
1818885-54-9
|
|
|
|
AR antagonist 1 is a potent antagonist of the androgen receptor. It binds to E3 ligase ligands with weak binding affinities to VHL protein in the synthesis of PR...
|
| T13187 |
Topterone
|
60607-35-4
|
100%
|
|
|
Topterone (Win 17,665) is a potent topical antiandrogen that inhibits the stimulation of lumbar organ development by testosterone and dihydrotestosterone in cast...
|
| T67818 |
BMS-641988
|
|
100%
|
|
|
BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer.
|
| T2991 |
3,3'-Diindolylmethane
|
1968-05-4
|
100%
|
|
|
3,3'-Diindolylmethane (DIM), a small molecule compound, is a proposed Y preventive agent.
|
| TN1805 |
Isosilybin B
|
142796-22-3
|
100%
|
|
|
Isosilybin B is a flavonolignan extracted from silymarin that exhibits anti-prostate cancer (PCA) activity, inhibits cancer cell proliferation, and contributes t...
|
| T8117 |
Metenolone acetate
|
434-05-9
|
100%
|
|
|
Metenolone acetate (Methenolone acetate) is an androgen and anabolic steroid (AAS) medication which is used mainly in the treatment of anemia due to bone marrow ...
|
