| T3390 |
Obacunone
|
751-03-1
|
98%
|
|
|
Obacunone has cytotoxicity in androgen-dependent human prostate Y cells. Obacunone exerts an antivirulence effect on S. Typhimurium and may serve as a lead compo...
|
| T0393 |
Anastrozole
|
120511-73-1
|
98%
|
|
|
Anastrozole (ZD1033)(ZD1033), a potent and highly selective aromatase (CYP19) inhibitor (IC50 = 15 nM), has no obvious effect on adrenocorticoid hormone synthesi...
|
| T7556 |
Fadrozole hydrochloride
|
102676-31-3
|
98%
|
|
|
Fadrozole hydrochloride (CGS 16949A) is a model aromatase inhibitor that has been shown to suppress estrogen production in the ovaries of fish.
|
| T1103 |
Aminoglutethimide
|
125-84-8
|
98%
|
|
|
Aminoglutethimide (BA-16038), an aromatase inhibitor, is used in the therapy of advanced BREAST Y.
|
| T3899 |
Calceolarioside B
|
105471-98-5
|
100%
|
|
|
Calceolarioside B (Desrhamnosyl isoacteoside) displays inhibition of aromatase. Calceolarioside B displays inhibition of human recombinant PKCalpha.
|
| T27320 |
Finrozole
|
160146-17-8
|
100%
|
|
|
Finrozole (MPV 2213ad) is a novel selective aromatase inhibitor that is partially reversible for breast development.
|
| T23549 |
YM 511
|
148869-05-0
|
100%
|
|
|
YM 511 is a highly specific non-steroidal aromatase inhibitor. YM 511 inhibits aromatase activities in microsomes from rat ovary and human placenta competitively...
|
| T26322L |
(-)-Vorozole
|
132042-69-4
|
97.14%
|
|
|
(-)-Vorozole is an orally active non-steroidal aromatase inhibitor with potency and selectivity. (-)-Vorozole has demonstrated antitumor activity in in vivo expe...
|
| T7197 |
Fadrozole
|
102676-47-1
|
98%
|
|
|
Fadrozole is a nonsteroidal aromatase inhibitor with potential antineoplastic activity(IC50 : 6.4 nM)
|
| T2O2744 |
Alpha-Naphthoflavone
|
604-59-1
|
98%
|
|
|
alpha-Naphthoflavone (7,8-benzoflavone), a synthetic flavonoid, is a potent inhibitor of aromatase with an I50 value of 0.5 μM.
|
| T71708 |
Minamestane
|
105051-87-4
|
99.04%
|
|
|
Minamestane is a novel irreversible aromatase inhibitor.Minamestane induces time-dependent inhibition of human placental aromatase with a half-life of 4 minutes ...
|
| T6917 |
Oleuropein
|
32619-42-4
|
99.16%
|
|
|
Oleuropein is an antioxidant polyphenol isolated from olive leaf.
|
| T27918 |
LY 43578
|
26766-35-8
|
99.62%
|
|
|
LY 43578 is an orally active aromatase inhibitor. LY43578 could inhibit O-demethylation of P-450-dependent p-nitroanisole and N-demethylation of ethylmorphine (I...
|
| T4281 |
Endoxifen
|
110025-28-0
|
99.66%
|
|
|
(E/Z)-Endoxifen ((E/Z)-Endoxifen) is an active metabolite of tamoxifen produced by the sequential action of cytochrome P450 (CYP) isoforms, including CYP2D6. It ...
|
| T1590 |
Letrozole
|
112809-51-5
|
99.68%
|
|
|
Letrozole (CGS 20267) is an Aromatase Inhibitor. The mechanism of action of letrozole is as an Aromatase Inhibitor.
|
| T1692 |
3-(3,4-Dimethoxyphenyl)propanoic acid
|
2107-70-2
|
99.68%
|
|
|
3-(3,4-Dimethoxyphenyl)propanoic acid (3,4-Dimethoxyhydrocinnamic acid) is an orally active short-chain fatty acid (SCFAs). It promotes γ-globin gene expression ...
|
| T1587 |
Exemestane
|
107868-30-4
|
99.73%
|
|
|
Exemestane (EXE) is an Aromatase Inhibitor. The mechanism of action of exemestane is as an Aromatase Inhibitor.
|
| T26322 |
Vorozole
|
129731-10-8
|
99.89%
|
|
|
Vorozole (R83842) is an orally active, potent, and selective nonsteroidal aromatase inhibitor.Vorozole exhibits antitumor activity in vivo and may be used in the...
|
| T0530 |
Flavanone
|
487-26-3
|
99.95%
|
|
|
Flavanone (2-Phenylchroman-4-one)s from citrus fruits have also been shown to exert beneficial effects on human vascular function. In particular, chronic interve...
|
| T12319 |
Org30958
|
99957-90-1
|
98%
|
|
|
Org30958 is a potent inhibitor of aromatase in vivo.
|
