| T6573 |
E 64c
|
76684-89-4
|
98%
|
|
|
E 64c (EP 475) , a derivative of E-64, is an irreversible and membrane-permeant cysteine protease inhibitor.
|
| T1080 |
2-Aminoethanethiol
|
60-23-1
|
98%
|
|
|
2-Aminoethanethiol (Cysteamine) is a Cystine Depleting Agent. The mechanism of action of cysteamine is as a Cystine Disulfide Reduction.
|
| T38469 |
(Rac)-Z-Phe-Phe-FMK
|
108005-94-3
|
98%
|
|
|
(Rac)-Z-Phe-Phe-FMK (Cathepsin L-IN-2) is a cathepsin L inhibitor that inhibits the tendency of β-amyloid to induce apoptotic changes .
|
| TP2056L |
Acetyl-Calpastatin (184-210)(human) acetate
|
|
98%
|
|
|
Acetyl-Calpastatin (184-210)(human) acetate is a potent, selective and reversible calpain inhibitor with Ki values of 0.2 nM and 6 μM for µ-calpain and cathepsin...
|
| T6035 |
Odanacatib
|
603139-19-1
|
98%
|
|
|
Odanacatib is an inhibitor of cathepsin K with potential anti-osteoporotic activity.
|
| T2493 |
PD 151746
|
179461-52-0
|
98%
|
|
|
PD151746 is a calpain inhibitor with a 20-fold selectivity for u-calpain (Ki = 0.26 ± 0.03 μM) over m-calpain (Ki = 5.33 ± 0.77 μM). Its IC50 values are 0.26 ± 0...
|
| T6037 |
E-64
|
66701-25-5
|
98%
|
|
|
E-64 (Proteinase inhibitor E 64) is an irreversible and specific cysteine protease inhibitor. The IC50 of E-64 for papain is 9 nM.
|
| T6432 |
Calpeptin
|
117591-20-5
|
98%
|
|
|
Calpeptin is a potent, cell-permeable calpain inhibitor.
|
| T37753 |
Aureusimine B
|
170713-71-0
|
98%
|
|
|
Aureusimine B, also known as phevalin, is a natural pyrazinone produced by certain fungi and by Staphylococcus spp., including S. aureus. Its synthesis appears t...
|
| T5211 |
NSC 185058
|
39122-38-8
|
98%
|
|
|
NSC 185058 is an inhibitor of ATG4B, a major cysteine protease. It also can attenuate the autophagic activity.
|
| T13911 |
Tacalcitol monohydrate
|
93129-94-3
|
98%
|
|
|
Tacalcitol monohydrate(Curatoderm monohydrate), a vitamin D3 analog that promotes bone development by regulating calcium ions, can be used to study psoriasis.
|
| T13288 |
VBY-825
|
1310340-58-9
|
98%
|
|
|
VBY-825 is a reversible inhibitor of cathepsin with high potency against cathepsins B, L, S and V.
|
| T6564 |
Leupeptin Hemisulfate
|
103476-89-7
|
98%
|
|
|
Leupeptin hemisulfate is a protease inhibitor with cell membrane-permeable, reversible, competitive, and oral activities. Leupeptin hemisulfate inhibits the acti...
|
| T19503 |
Papain
|
9001-73-4
|
|
|
|
Papain is a cysteine protease of the peptidase C1 family. Papain is used in food, pharmaceutical, textile, and cosmetic industries.
|
| T2470 |
MDL-28170
|
88191-84-8
|
|
|
|
MDL-28170 (Calpain Inhibitor III) is a Cysteine protease.
|
| T0448 |
(S)-(+)-Ibuprofen
|
51146-56-6
|
100%
|
|
|
(S)-(+)-Ibuprofen (Dexibuprofen) , is a non-steroidal anti-inflammatory drug (NSAID), inhibiting cyclooxygenase (COX).
|
| T16089 |
MK-0674
|
887781-62-6
|
100%
|
|
|
MK-0674 is an orally available, selective and potent cathepsin K inhibitor (IC50: 0.4 nM) that inhibits Cat B, Cat F, Cat L, and Cat S. It can be used in metabol...
|
| T3420 |
CA-074 methyl ester
|
147859-80-1
|
97.26%
|
|
|
CA-074 methyl ester (Cathepsin B Inhibitor IV) is a specific inhibitor of Cathepsin B with neuroprotective, anti-cancer, and anti-inflammatory effects.
|
| T1850 |
Balicatib
|
354813-19-7
|
97.78%
|
|
|
Balicatib (AAE581) is a potent and selective inhibitor of cathepsin K, used in trials studying the treatment of osteoporosis.
|
| T21509 |
CA 074
|
134448-10-5
|
97.80%
|
|
|
CA 074 is a potent inhibitor of cathepsin B with a Ki value of 2 to 5 nM.CA 074 inhibits ischemic hippocampal neuronal death in primates and attenuates retinopat...
|
