| T20625 |
Prochloraz
|
67747-09-5
|
98%
|
|
|
Prochloraz (Prelude) is a broad-spectrum contact imidazole fungicide. Prochloraz inhibits human placental microsomal aromatase in vitro (IC50 = 40 nM). Prochlora...
|
| T13542 |
α-Zearalenol
|
36455-72-8
|
98%
|
|
|
α-Zearalenol is one of the major metabolites of Zearalenone. α-Zearalenol has structural analogy to estrogen, thus α-Zearalenol can bind to estrogen receptors (E...
|
| TN1567 |
Delphinidin chloride
|
528-53-0
|
98%
|
|
|
Delphinidin chloride, a natural plant pigment found in berries and red wine, is a precursor of certain anthocyanins. Delphinidin chloride induces the release of ...
|
| T21897L |
MPP hydrochloride
|
|
98%
|
|
|
MPP hydrochloride is a selective estrogen receptor (ERR) modulator.
|
| T6743 |
(E/Z)-4-Hydroxytamoxifen
|
68392-35-8
|
|
|
|
(E/Z)-4-Hydroxytamoxifen (Afimoxifene) is the active metabolite of tamoxifen and a selective estrogen receptor (ER) modulator that is widely used in the therapeu...
|
| T5633 |
H3B-5942
|
2052128-15-9
|
|
|
|
H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).
|
| T7389 |
G15
|
1161002-05-6
|
|
|
|
G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)
|
| T1424 |
Ethynyl estradiol
|
57-63-6
|
100%
|
|
|
Ethynyl estradiol is a semisynthetic alkylated ESTRADIOL with a 17-alpha-ethinyl substitution. It has high estrogenic potency when administered orally, and is of...
|
| T3846 |
Bavachin
|
19879-32-4
|
100%
|
|
|
Bavachin (Corylifolin) is a phytoestrogen that activates the estrogen receptors ERα and ERβ.
|
| T1579 |
Mestranol
|
72-33-3
|
100%
|
|
|
Mestranol (Devocin), a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.
|
| T3645 |
Endoxifen E-isomer hydrochloride
|
1197194-61-8
|
96.47%
|
|
|
Endoxifen E-isomer hydrochloride (E-Endoxifen hydrochloride) , a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
|
| T2250 |
DY131
|
95167-41-2
|
96.72%
|
|
|
DY131 (DY-131) is a novel selective agonist of ERRβ and ERRγ.
|
| T0035 |
Dienestrol
|
84-17-3
|
96.73%
|
|
|
Dienestrol (Restrol) is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist. Estrogens can increase a normal clear discharge from the va...
|
| T1571 |
Estriol
|
50-27-1
|
97.48%
|
|
|
Estriol (Oestriol) is a hydroxylated metabolite of ESTRADIOL or ESTRONE that has a hydroxyl group at C3, 16-alpha, and 17-beta position. Estriol is a major urina...
|
| TN1768 |
Iriflophenone
|
52591-10-3
|
97.53%
|
|
|
Iriflophenone stimulates cells proliferation in MCF-7 and T-47D human breast cancer.
|
| T8370 |
GSK5182
|
877387-37-6
|
97.63%
|
|
|
GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)
|
| T2882 |
Genistin
|
529-59-9
|
97.65%
|
|
|
Genistin (Genistoside) is the major isoflavonoid of soybeans and soy products.It has been reported to possess various therapeutic effects, including anti-inflamm...
|
| T15788 |
LSZ-102
|
2135600-76-7
|
97.84%
|
|
|
LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.
|
| T5S0543 |
Isocurcumenol
|
24063-71-6
|
98%
|
|
|
1. Isocurcumenol inhibits 5α-reductase which converts testosterone to dihydrotestosterone (DHT).
|
| T2544 |
Bazedoxifene acetate
|
198481-33-3
|
98%
|
|
|
Bazedoxifene acetate (WAY-TES 424) is a novel selective estrogen receptor modulator (SERM).
|
