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Estrogen/progestogen Receptor

Estrogen receptors are a group of proteins found inside cells. They are receptors that are activated by the hormone estrogen (17β-estradiol). Two classes of estrogen receptor exist: ER, which is a member of the nuclear hormone family of intracellular receptors, and GPER (GPR30), which is a member of the rhodopsin-like family of G protein-coupled receptors.The progesterone receptor (PR), also known as NR3C3 or nuclear receptor subfamily 3, group C, member 3, is a protein found inside cells. It is activated by the steroid hormone progesterone.
Cat. No. 製品名 CAS No. Purity Chemical Structure
T26537 AC-186 1421854-16-1 98%
AC-186 is a nonsteroidal estrogen receptor β (ERβ) agonist with different affinities for ERβ and ERα, with an EC50 of 6 nM for ERβ and 5000 nM for ERα. AC-186 ha...
T77577 SLU-PP-332 303760-60-3 98%
SLU-PP-332 is a pan-estrogen receptor-related receptor (ERR) agonist with high affinity for ERRα, ERRβ, and ERRγ with EC50 values of 98, 230, and 430 nM, respect...
T1490 Gestodene 60282-87-3 98%
Gestodene (WL 70) is a progestogen hormonal contraceptive.
T6743 (E/Z)-4-Hydroxytamoxifen 68392-35-8
(E/Z)-4-Hydroxytamoxifen (Afimoxifene) is the active metabolite of tamoxifen and a selective estrogen receptor (ER) modulator that is widely used in the therapeu...
T20720 Norethisterone enanthate 3836-23-5
Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects.
T5633 H3B-5942 2052128-15-9
H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).
T4505 Ferrous Bisglycinate 20150-34-9
Ferrous Bisglycinate (Bisglycine iron(II) salt) is used in the fortification of infant formulations and foods.
T3399 Psoralidin 18642-23-4
Psoralidin inhibits Akt phosphorylation and phosphatidylinositol 3-kinase activation and transcriptionally. Psoralidin possesses anticancer and chemopreventive p...
T5040 Medroxyprogesterone 520-85-4
Medroxyprogesterone is used in the treatment of renal carcinoma. It is a synthetic progestational hormone used in veterinary practice as an estrus regulator.
T1536 Promestriene 39219-28-8
Promestriene (3-propyl ethyl) (INN) is a synthetic estrogen and glucocorticoid used topically in a 1% cream formulation. It is described as a tropic agent and an...
T1424 Ethynyl estradiol 57-63-6 100%
Ethynyl estradiol is a semisynthetic alkylated ESTRADIOL with a 17-alpha-ethinyl substitution. It has high estrogenic potency when administered orally, and is of...
T11230 ERRα antagonist-1 1072145-33-5 100%
ERRα antagonist-1 (ERR+/- antagonist-1) is a high-affinity, selective antagonist of the estrogen-related receptor α (ERRα). It effectively prevents the interacti...
T3846 Bavachin 19879-32-4 100%
Bavachin (Corylifolin) is a phytoestrogen that activates the estrogen receptors ERα and ERβ.
T1579 Mestranol 72-33-3 100%
Mestranol (Devocin), a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.
T13675 Elacestrant dihydrochloride 1349723-93-8 100%
Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ERα and 870 nM for ER...
T9799 Serba-2 533884-08-1 100%
Serba-2 is an agonist of benzopyran selective estrogen receptor beta.
T1438 Butoconazole nitrate 64872-77-1 100%
Butoconazole Nitrate is the nitrate salt form of butoconazole, a synthetic imidazole derivative with fungistatic properties. Butoconazole nitrate (RS 35887) inte...
T2559 Allylestrenol 432-60-0 100%
Allylestrenol (Gestanin) is a synthetic steroid with progestational activity.
T9800 Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- 533883-77-1 95.18%
Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- is an estrogen receptor beta (ERβ) agonist.
T3645 Endoxifen E-isomer hydrochloride 1197194-61-8 96.47%
Endoxifen E-isomer hydrochloride (E-Endoxifen hydrochloride) , a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
AC-186
T26537
AC-186 is a nonsteroidal estrogen receptor β (ERβ) agonist with different affinities for ERβ and ERα, with an EC50 of 6 nM for ERβ and 5000 nM for ERα. AC-186 ha...
SLU-PP-332
T77577
SLU-PP-332 is a pan-estrogen receptor-related receptor (ERR) agonist with high affinity for ERRα, ERRβ, and ERRγ with EC50 values of 98, 230, and 430 nM, respect...
Gestodene
T1490
Gestodene (WL 70) is a progestogen hormonal contraceptive.
(E/Z)-4-Hydroxytamoxifen
T6743
(E/Z)-4-Hydroxytamoxifen (Afimoxifene) is the active metabolite of tamoxifen and a selective estrogen receptor (ER) modulator that is widely used in the therapeu...
Norethisterone enanthate
T20720
Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects.
H3B-5942
T5633
H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).
Ferrous Bisglycinate
T4505
Ferrous Bisglycinate (Bisglycine iron(II) salt) is used in the fortification of infant formulations and foods.
Psoralidin
T3399
Psoralidin inhibits Akt phosphorylation and phosphatidylinositol 3-kinase activation and transcriptionally. Psoralidin possesses anticancer and chemopreventive p...
Medroxyprogesterone
T5040
Medroxyprogesterone is used in the treatment of renal carcinoma. It is a synthetic progestational hormone used in veterinary practice as an estrus regulator.
Promestriene
T1536
Promestriene (3-propyl ethyl) (INN) is a synthetic estrogen and glucocorticoid used topically in a 1% cream formulation. It is described as a tropic agent and an...
Ethynyl estradiol
T1424
Ethynyl estradiol is a semisynthetic alkylated ESTRADIOL with a 17-alpha-ethinyl substitution. It has high estrogenic potency when administered orally, and is of...
ERRα antagonist-1
T11230
ERRα antagonist-1 (ERR+/- antagonist-1) is a high-affinity, selective antagonist of the estrogen-related receptor α (ERRα). It effectively prevents the interacti...
Bavachin
T3846
Bavachin (Corylifolin) is a phytoestrogen that activates the estrogen receptors ERα and ERβ.
Mestranol
T1579
Mestranol (Devocin), a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.
Elacestrant dihydrochloride
T13675
Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ERα and 870 nM for ER...
Serba-2
T9799
Serba-2 is an agonist of benzopyran selective estrogen receptor beta.
Butoconazole nitrate
T1438
Butoconazole Nitrate is the nitrate salt form of butoconazole, a synthetic imidazole derivative with fungistatic properties. Butoconazole nitrate (RS 35887) inte...
Allylestrenol
T2559
Allylestrenol (Gestanin) is a synthetic steroid with progestational activity.
Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-
T9800
Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- is an estrogen receptor beta (ERβ) agonist.
Endoxifen E-isomer hydrochloride
T3645
Endoxifen E-isomer hydrochloride (E-Endoxifen hydrochloride) , a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
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