T1325 |
Carprofen
|
53716-49-7
|
98%
|
|
Carprofen (Ridamyl) is a propionic acid derivate and nonsteroidal anti-inflammatory drug (NSAID) with anti-inflammatory, analgesic, and antipyretic activities.
|
T28353 |
PDP-EA
|
861891-72-7
|
98%
|
|
PDP-EA is an activator of fatty acid amide hydrolase(FAAH) and enhances the amidohydrolase activity of FAAH.
|
T23119 |
Palmitoylisopropylamide
|
189939-61-5
|
98%
|
|
Palmitoylisopropylamide is a selective FAAH inhibitor that inhibits [H]-AEA uptake and cell proliferation at low concentrations.
|
T4323 |
PF-04457845
|
1020315-31-4
|
98%
|
|
PF-04457845 is a greatly and effctive FAAH inhibitor, and for hFAAH(IC50=7.2±0.63 nM) and rFAAH(IC50=7.4±0.62 nM).
|
TN1965 |
N-Benzyllinolenamide
|
883715-18-2
|
98%
|
|
N-Benzyllinolenamide is a natural product. It is an inhibitor of fatty acid amide hydrolase (FAAH, IC50 of 41.8 μM).
|
T3S2105 |
N-Benzylpalmitamide
|
74058-71-2
|
98%
|
|
N-Benzylpalmitamide (Macamide 1) inhibits fatty acid amide hydrolase (FAAH) in a time-dependent manner and could potentially offer a good alternative for the tre...
|
T67896 |
CB2R/FAAH modulator-1
|
928892-60-8
|
100%
|
|
CB2R/FAAH modulator-1, a cannabinoid type 2 receptor (CB2R) agonist, is also a fatty acid amide hydrolase (FAAH) inhibitor (IC50=4 μM) that reduces the productio...
|
T2859 |
Biochanin A
|
491-80-5
|
97.1%
|
|
Biochanin A (4-Methylgenistein) is an isoflavone derivative isolated from red clover Trifolium pratense with anticarcinogenic properties. Biochanin A is a natura...
|
T6714 |
URB-597
|
546141-08-6
|
97.84%
|
|
URB-597 (FAAH Inhibitor II) is an effective, orally bioavailable FAAH inhibitor (IC50: 4.6 nM), and no effect on other cannabinoid-related targets.
|
T6043 |
PF-3845
|
1196109-52-0
|
98%
|
|
PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2.
|
T11256 |
FAAH inhibitor 1
|
326866-17-5
|
98.05%
|
|
FAAH inhibitor 1 (Benzothiazole analog 3) is an effective FAAH inhibitor with an IC50 of 18 nM.
|
T15802 |
LY2183240
|
874902-19-9
|
98.17%
|
|
LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 27...
|
T5357 |
ARN272
|
488793-85-7
|
98.23%
|
|
ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).
|
T68492 |
AM 374
|
86855-26-7
|
98.39%
|
|
AM 374 (HDSF) is an fatty acid amide hydrolase (FAAH) inhibitor. AM 374 inhibits amidase activity with an IC 50 value of 13 nM. AM 374 can be used for the resear...
|
T16515 |
PF 750
|
959151-50-9
|
98.83%
|
|
PF 750 (ZINC27647189) is a selective and covalent inhibitor of FAAH. PF 750 shows IC50s varying from 16.2 to 595 nM in different incubation times.
|
T67747 |
CB2R/FAAH modulator-3
|
2876918-67-9
|
99.02%
|
|
CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH. CB2R/FAAH modulator-3 acts as a CB2R agonist and FAAH inhibitor, the Ki values are...
|
T7688 |
4-Nonylphenylboronic acid
|
256383-45-6
|
99.13%
|
|
4-Nonylphenylboronic acid is a inhibitor of FAAH.
|
T15268 |
FAAH-IN-2
|
184475-71-6
|
99.18%
|
|
FAAH-IN-2 (O-Desmorpholinopropyl Gefitinib) is a potent inhibitor of FAAH(fatty acid amide hydrolase).
|
T77594 |
VU534
|
923509-20-0
|
99.22%
|
|
VU534 is a NAPE-PLD agonist with an EC50 of 0.30 μM.VU534 is a dual inhibitor of FAAH and sEH, with an IC50 of 1.2 μM for sEH.VU534 is used in diseases related t...
|
T77513 |
2-Chlorophenylboronic acid
|
3900-89-8
|
99.42%
|
|
2-Chlorophenylboronic acid is a monohalogenated phenylboronic acid, which is an important pharmaceutical intermediate and is widely used in the synthesis of new ...
|