| T21793 |
CGP 35348
|
123690-79-9
|
98%
|
|
|
CGP 35348 is a selective antagonist of GABAB receptor (EC50 = 34 μM). CGP 35348 can be used in studies of neuromuscular coordination and spatial learning after n...
|
| T28479 |
PZ-II-029
|
164025-44-9
|
98%
|
|
|
PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.
|
| TMS0418 |
Dihydroergotoxine mesylate
|
8067-24-1
|
98%
|
|
|
Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.
|
| T16539 |
Piperazine citrate
|
144-29-6
|
98%
|
|
|
Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring. It used as an Anthelmi...
|
| T8268 |
6,2'-Dihydroxyflavone
|
92439-20-8
|
98%
|
|
|
6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.
|
| T32098L |
Homocarnosine acetate
|
|
98%
|
|
|
Homocarnosine acetate is a dipeptide unique to brain consisting of γ-aminobutyric acid (GABA) and histidine. Homocarnosine acetate has antioxidant and anti-infla...
|
| T37190 |
L-Allylglycine
|
16338-48-0
|
98%
|
|
|
L-Allylglycine is an amino acid derivative that reduces glutamate decarboxylase (GAD) activity by 60% when administered at a dose of 39.8 μmol/g per hour ex vivo...
|
| T1240 |
Flumazenil
|
78755-81-4
|
98%
|
|
|
Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervous ...
|
| TQ0151 |
L-655708
|
130477-52-0
|
98%
|
|
|
L-655708 is a selective and highly potent GABAA receptor reverse agonist with a Ki value of 0.45 nM.
|
| T3173 |
DAA-1106
|
220551-92-8
|
98%
|
|
|
DAA-1106 is a potent and selective ligand for peripheral benzodiazepine receptor (PBR), acting as a potent and selective agonist at the peripheral benzodiazepine...
|
| T3644 |
U93631
|
152273-12-6
|
98%
|
|
|
GABAA receptor antagonist that binds the picrotoxin site and stabilizes the inactive form of the channel via allosteric interaction. Accelerates the decay of GAB...
|
| T4993 |
Afloqualone
|
56287-74-2
|
98%
|
|
|
Afloqualone (HQ-495) is a agonist of GABA Receptor . Target: GABA Receptor in vitro: Afloqualone is a quinazolinone family GABAergic drug. It has sedative and mu...
|
| T2067 |
NS11394
|
951650-22-9
|
98%
|
|
|
NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(1...
|
| TN1308 |
6-Hydroxyflavanone
|
4250-77-5
|
98%
|
|
|
6-Hydroxyflavanone, extracted from the leaves of Acorus calamus, exhibits anti-inflammatory and anti-neuropathic pain activity by targeting cyclooxygenase-2 (COX...
|
| T5330 |
Fluralaner
|
864731-61-3
|
98%
|
|
|
Fluralaner (A1443) is an isoxazoline ectoparasiticide. It potently and selectively inhibits binding of the GABA receptor channel blocker EBOB to housefly head me...
|
| TN1023 |
Miltirone
|
27210-57-7
|
98%
|
|
|
Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.
|
| T24381 |
L-822179
|
215874-86-5
|
98%
|
|
|
L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.
|
| T16489 |
Darigabat
|
1614245-70-3
|
98%
|
|
|
Darigabat (PF-06372865) is an orally active and selective GABAA receptor modulator that crosses the blood-brain barrier and exhibits anxiolytic activity, with Ki...
|
| T77796 |
DL-Borneol
|
507-70-0
|
98%
|
|
|
DL-Borneol ((endo)-Borneol) is a small molecule extracted from traditional Chinese medicine (TCM). It is an orally bioadjuvant that improves drug delivery to the...
|
| T22813 |
GS 39783
|
39069-52-8
|
98%
|
|
|
GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement and condition...
|
