| T22986 |
MK 1903
|
1268882-43-4
|
98%
|
|
|
MK 1903 is a potent and selective complete agonist for the hydroxy-carboxylic acid receptor 2 (HCA2). HCA2 is also known as G protein-coupled receptor 109A(GPR10...
|
| TN1849 |
Kuwanon H
|
76472-87-2
|
98%
|
|
|
Kuwanon H, and possibly kuwanon G also, are specific antagonists for the gastrin-releasing peptide (GRP) -preferring receptor and can be useful for studying the ...
|
| T12216 |
NF-56-EJ40
|
2380230-73-7
|
98%
|
|
|
NF-56-EJ40 is an effective and highly selective antagonist of human SUCNR1 with an IC50 of 25 nM and a Ki of 33 nM.
|
| TP1345 |
Kisspeptin-10, human (TFA)(374675-21-5,FREE)
|
TP1345
|
98%
|
|
|
Kisspeptin-10, human TFA is a potent vasoconstrictor and angiogenesis inhibitor. Kisspeptin-10, human TFA acts as a tumor metastasis suppressor via its receptor ...
|
| T1793 |
MBX-2982
|
1037792-44-1
|
98%
|
|
|
MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.
|
| T1781 |
GW9508
|
885101-89-3
|
98%
|
|
|
GW9508(GW 9508) is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in a glucose-sensitive manner.
|
| T15413 |
GPR120 Agonist 3
|
1599477-75-4
|
98%
|
|
|
GPR120 Agonist 3 (GPR120-IN-1) is a selective agonist of Gpr120 ( logEC50: -7.62).
|
| TP1928L1 |
[Orn5]-URP acetate
|
TP1928L1
|
98%
|
|
|
[Orn5]-URP acetate is an effective and selective Urotensin-II receptor (UT) antagonist (pEC50 = 7.24). [Orn5]-URP exhibits no agonist activity.
|
| T37526 |
2-Oleoylglycerol
|
3443-84-3
|
98%
|
|
|
2-Oleoylglycerol is a lipid found in palm kernel, sunflower seed and rice bran.2-Oleoylglycerol acts as a GPR119 agonist with neuroprotective effects and induces...
|
| T83972 |
NOX-6-18
|
898211-21-7
|
98%
|
|
|
NOX-6-18 (GPR132-B-160) is a highly potent and selective GPR132 antagonist with insulinotropic activity that modulates macrophage reprogramming in pancreatic isl...
|
| T60074 |
GPCR agonist-2
|
291528-35-3
|
98%
|
|
|
GPCR agonist-2 (4-(Cyclopropylamino)-3-nitrobenzoic acid) is an agonist of the orphan human GPCR GPR109B.
|
| T5351L |
PU-WS13 hydrobromide
|
|
98%
|
|
|
PU-WS13 hydrobromide is a GRP94 inhibitor with anti-inflammatory activity and inhibits the proliferation of M2-like macrophages in mouse TNBC tumors.
|
| T36036 |
CAY10786
|
1239987-91-7
|
98%
|
|
|
CAY10786 (GPR52 antagonist-1) is an antagonist of G protein-coupled receptor 52 (GPR52, IC50 = 0.63 μM).
|
| T7359 |
CAY10471 Racemate
|
844639-57-2
|
|
|
|
CAY10471 Racemate (TM30089 Racemate) is a potent, highly selective CRTH2/DP 2 receptor antagonist. CAY10471 Racemate binds to the human CRTH2/DP2, DP1, and TP re...
|
| T1286 |
Vincamine
|
1617-90-9
|
|
|
|
Vincamine (Perval) is a major alkaloid of Vinca minor L., Apocynaceae. It has been used therapeutically as a vasodilator and antihypertensive agent, particularly...
|
| T7127 |
DC260126
|
346692-04-4
|
|
|
|
DC260126 is a small-molecule antagonist of FFA1 (GPR40)
|
| T5406 |
SNAP 94847
|
487051-12-7
|
|
|
|
SNAP 94847 (SNAP-94847) is a selective and competitive MCH1 receptor (MCH1-R) antagonist (Ki: 2.2 nM). It has anxiolytic and antidepressant activity and reduces ...
|
| T2351 |
Fasiglifam
|
1000413-72-8
|
|
|
|
Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.
|
| T36818 |
Questiomycin A
|
1916-59-2
|
|
|
|
Questiomycin A is an antibiotic produced in crème fraiche with antibacterial and anticancer activities. Questiomycin A suppresses expression of GRP78, a cell-pro...
|
| T12095 |
Monomethyl fumarate
|
2756-87-8
|
|
|
|
Monomethyl fumarate is a potent agonist of GPR109A .
|
