| T0185 |
Escitalopram
|
128196-01-0
|
94.62%
|
|
|
Escitalopram (Seroplex) is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing e...
|
| T40652 |
Meclizine
|
569-65-3
|
95.16%
|
|
|
Meclizine, also known as Meclozine, is a piperazine class H1 antagonist with antihistamine properties that inhibits the interaction of histamine at H1 receptors ...
|
| T0445L |
Promethazine hydrochloride
|
58-33-3
|
95.36%
|
|
|
Promethazine hydrochloride (Promethazine HCl) , the first-generation antihistamine, is a strong antagonist of the H1 receptor and a moderate antagonist of the mA...
|
| TQ0046 |
Bavisant
|
929622-08-2
|
96.06%
|
|
|
Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist. Bavisant can be used in research on mechanisms of action, involving wakefu...
|
| T68122L |
Oxmetidine FA
|
|
96.48%
|
|
|
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.
|
| T13566 |
Bamirastine
|
215529-47-8
|
96.68%
|
|
|
Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on alle...
|
| T3979 |
Emedastine
|
87233-61-2
|
97.1%
|
|
|
Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. Emedastine reversibly and competitively blo...
|
| T79499 |
KSK68
|
2566715-91-9
|
97.22%
|
|
|
KSK68 is a potent dual sigma-1 and histamine H3 receptor antagonist with potential analgesic activity and high affinity for H3 receptors, sigma-1, sigma-2 recept...
|
| T19443 |
N-Acetylhistamine
|
673-49-4
|
97.72%
|
|
|
N-Acetylhistamine (N-Omega-acetylhistamine) is a metabolite of histamine.
|
| T13352 |
Wy 49051
|
113418-56-7
|
97.9%
|
|
|
Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).
|
| T4196 |
Betahistine EP Impurity C
|
5452-87-9
|
98%
|
|
|
Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.
|
| T7524 |
Metiamide
|
34839-70-8
|
98%
|
|
|
Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .
|
| T7413 |
JNJ-5207852
|
398473-34-2
|
98%
|
|
|
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
|
| T1182 |
Levocarnitine propionate hydrochloride
|
119793-66-7
|
98%
|
|
|
Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, intermittent claudica...
|
| T20884 |
Hydroxyzine
|
68-88-2
|
98%
|
|
|
Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.
|
| T1030 |
Triprolidine hydrochloride monohydrate
|
6138-79-0
|
98%
|
|
|
Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.
|
| T11723L |
JNJ-39758979
|
1046447-90-8
|
98.00%
|
|
|
JNJ-39758979 is a selective and high-affinity histamine H4 receptor antagonist (Kis: 12.5, 5.3, and 25 nM for human, mouse, and monkey histamine H4 receptor, res...
|
| T1393 |
Sodium butanoate
|
156-54-7
|
98.02%
|
|
|
Sodium butanoate (Sodium Butyrate) is the sodium salt of butyrate with potential antineoplastic activity. Butyrate, a short chain fatty acid, competitively binds...
|
| T1045 |
Trimipramine maleate
|
521-78-8
|
98.02%
|
|
|
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepineph...
|
| TQ0066 |
GSK189254A
|
720690-73-3
|
98.04%
|
|
|
GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).
|
