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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Cat. No. 製品名 CAS No. Purity Chemical Structure
T3723 Dioxopromethazine hydrochloride 15374-15-9 99%
Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
TN1008 Psoralenoside 905954-17-8 99.03%
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activi...
T10680 Carebastine 90729-42-3 99.06%
Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
T17072 Thiethylperazine dimaleate 1179-69-7 99.07%
Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor. Thiethylperazine dimaleate is an activator of ABCC1 an...
T1110 Meclizine dihydrochloride 1104-22-9 99.08%
Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation si...
T9770 Samelisant 1394808-82-2 99.09%
Samelisant (SUVN-G3031) is a selective and inverse agonist of H3 receptor with Kis of 8.7 nM and 9.8 nM for human and rat. Samelisant has anticataplectic effects...
T8548 Metoprine 7761-45-7 99.09%
Metoprine is a potent inhibitor of histamine N-methyltransferase (HMT), with potential antineoplastic activity.
T12489 Pimethixene 314-03-4 99.1%
Pimethixene (Calmixen) is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist...
T3610 Ranitidine 66357-35-5 99.1%
Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors). It is used to treat gastrointestina...
T10499 H3 receptor-MO-1 1240914-03-7 99.11%
H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.
T0445 Promethazine 60-87-7 99.11%
Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
T68056 Donetidine 99248-32-5 99.12%
Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
T0865 Ranitidine Hydrochloride 66357-59-3 99.13%
Ranitidine Hydrochloride (AH19065) is a member of the class of histamine H2-receptor antagonists with antacid activity. Ranitidine is a competitive and reversibl...
T15005 CP-66948 101189-47-3 99.14%
CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.
T4087 S 38093 HCl 1222097-72-4 99.16%
S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.
T0074L Chlorprothixene hydrochloride 6469-93-8 99.16%
Chlorprothixene hydrochloride (Truxal hydrochloride) brings strong blocking effects by blocking the 5-HT2 D1, D2, D3, histamine H1, muscarinic and alpha1 adrener...
T22501 2-Pyridylethylamine dihydrochloride 3343-39-3 99.17%
2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.
T0383 Fenspiride hydrochloride 5053-08-7 99.18%
Fenspiride hydrochloride (Decaspiride) , an oxazolidinone spiro compound, is a drug used in the therapy of certain respiratory diseases. It is approved for use i...
T68100 Mifentidine 83184-43-4 99.20%
Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.
T0059 Diphenylpyraline hydrochloride 132-18-3 99.22%
Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) is used in the treatment of Parkinsonism.It is a first-generation antihistami...
Dioxopromethazine hydrochloride
T3723
Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
Psoralenoside
TN1008
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activi...
Carebastine
T10680
Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
Thiethylperazine dimaleate
T17072
Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor. Thiethylperazine dimaleate is an activator of ABCC1 an...
Meclizine dihydrochloride
T1110
Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation si...
Samelisant
T9770
Samelisant (SUVN-G3031) is a selective and inverse agonist of H3 receptor with Kis of 8.7 nM and 9.8 nM for human and rat. Samelisant has anticataplectic effects...
Metoprine
T8548
Metoprine is a potent inhibitor of histamine N-methyltransferase (HMT), with potential antineoplastic activity.
Pimethixene
T12489
Pimethixene (Calmixen) is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist...
Ranitidine
T3610
Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors). It is used to treat gastrointestina...
H3 receptor-MO-1
T10499
H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.
Promethazine
T0445
Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
Donetidine
T68056
Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
Ranitidine Hydrochloride
T0865
Ranitidine Hydrochloride (AH19065) is a member of the class of histamine H2-receptor antagonists with antacid activity. Ranitidine is a competitive and reversibl...
CP-66948
T15005
CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.
S 38093 HCl
T4087
S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.
Chlorprothixene hydrochloride
T0074L
Chlorprothixene hydrochloride (Truxal hydrochloride) brings strong blocking effects by blocking the 5-HT2 D1, D2, D3, histamine H1, muscarinic and alpha1 adrener...
2-Pyridylethylamine dihydrochloride
T22501
2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.
Fenspiride hydrochloride
T0383
Fenspiride hydrochloride (Decaspiride) , an oxazolidinone spiro compound, is a drug used in the therapy of certain respiratory diseases. It is approved for use i...
Mifentidine
T68100
Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.
Diphenylpyraline hydrochloride
T0059
Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) is used in the treatment of Parkinsonism.It is a first-generation antihistami...
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