ペプチド
抗体
色素試薬
PROTAC
バーチャルスクリーニング
TargetMolキット
Cell Counting Kit-8 (CCK-8)
Inhibitor Cocktails
天然化合物
フェノール類
アルカロイド類
フラボノイド類
阻害剤
血管新生
アポトーシス
オートファジー
細胞周期・チェックポイント
クロマチン・エピジェネティック
細胞骨格シグナル
DNA損傷・DNA修復
内分泌・ホルモン
GPCR/Gタンパク質
免疫・炎症
JAK・STATシグナル
| Cat. No. | 製品名 | CAS No. | Purity | Chemical Structure |
|---|---|---|---|---|
| T3257 | UNC0638 | 1255580-76-7 | 98% |
|
| UNC0638 is an inhibitor of β-protein lysine methyltransferases G9a(IC50<15 nM) and GLP(IC50=19 nM) with excellent potency and selectivity over a wide range of ep... | ||||
| T28036 | MI-2-2 | 1454920-20-7 | 98% |
|
| MI-2-2 is an inhibitor of bivalent protein-protein interaction between menin and MLL with an IC50 of 46 nM. MI-2-2 binds to menin with Kd of 22 nM. | ||||
| T4393 | MS049 2HCl (1502816-23-0(free base)) | T4393 | 98% |
|
| MS049 is a potent and selective inhibitor of PRMT4 (IC50 = 34 nM) and PRMT6 (IC50 = 43 nM). It is less active against additional type I PRMTs (IC50s = >130, >220... | ||||
| T5322 | BCI-121 | 432529-82-3 | 98% |
|
| BCI-121 is a substrate-competitive SMYD3 inhibitor that inhibits the proliferation of the cancer cell. | ||||
| T0174 | Cyproheptadine hydrochloride sesquihydrate | 41354-29-4 | 98% |
|
| Cyproheptadine hydrochloride sesquihydrate, an antihistamine, is an antagonist of serotonin and histamine2. | ||||
| T3084 | SGC707 | 1687736-54-4 | 98% |
|
| SGC707 is a potent, selective, and cell-active allosteric inhibitor of PRMT3. | ||||
| T6803 | Chaetocin | 28097-03-2 | 98% |
|
| Chaetocin, a natural product from Chaetomium species, is a histone methyltransferase inhibitor with IC50 of 0.8 μM, 2.5 μM and 3 μM for dSU(VAR)3-9, mouse G9a an... | ||||
| T16886 | Sinefungin | 58944-73-3 | 98% |
|
| Sinefungin is an effective inhibitor of virion mRNA(guanine-7-)-methyltransferase, mRNA(nucleoside-2'-)-methyltransferase, and viral multiplication. Sinefungin i... | ||||
| T36798 | SW2_110A | 2579696-95-8 | 98% |
|
| SW2_110A is a cell-permeable, selective chromosome group 8 chromosome domain (CBX8 ChD) inhibitor with a Kd of 800 nM. In vitro, SW2_110A is 5-fold more selectiv... | ||||
| T15194 | EBI-2511 | 2098546-05-3 | 98% |
|
| EBI-2511 is a highly potent and orally active inhibitor of EZH2 (IC50: 6 nM in Pfeffiera cell lines). | ||||
| T6879 | LLY-507 | 1793053-37-8 | 98% |
|
| LLY-507 is an effective, cell-active, and specific inhibitor of protein-lysine Methyltransferase SMYD2. | ||||
| T13954 | UNC6852 | 2688842-08-0 | 98% |
|
| UNC6852 contains an EED ligand (IC50 = 247 nM) and a von Hippel-Lindau ligand and is a selective polycomb repressive complex 2 (PRC2) degrader based on PROTAC. | ||||
| T2097 | C-7280948 | 587850-67-7 | 98% |
|
| C-7280948 is a PRMT1 inhibitor. | ||||
| T4021 | UNC3866 | 1872382-47-2 | 98% |
|
| UNC3866 is a potent antagonist of the CBX7-H3 interaction as determined by AlphaScreen. | ||||
| T9584 | UNC6934 | 2561494-77-5 | 98% |
|
| UNC6934 is a chemical probe targeting the N-terminal PWWP (PWWP1) domain of NSD2. | ||||
| T2354 | UNC 0631 | 1320288-19-4 | 98% |
|
| UNC0631 is a effectvie histone methyltransferase G9a inhibitor (IC50=4 nM). | ||||
| T8879 | MR837 | 1210906-48-1 | 98% |
|
| ZINC30303842 is a NSD2-PWWP1 antagonist. | ||||
| T4021L | UNC3866 TFA(1872382-47-2 free base) | 1872382-48-3 | 98% |
|
| UNC3866 TFA is a potent antagonist of the CBX7-H3 interaction as determined by AlphaScreen. | ||||
| T1905 | EPZ005687 | 1396772-26-1 | 98% |
|
| EPZ005687 is a potent and selective inhibitor of EZH2. | ||||
| T2643 | MI-3 | 1271738-59-0 | 98% |
|
| MI-3 (Menin-MLL Inhibitor) is an effective inhibitor of Menin-MLL interaction (IC50: 648 nM). | ||||
