| T11966 |
MCHR1 antagonist 2
|
863115-70-2
|
98%
|
|
|
MCHR1 antagonist 2 is an antagonist of melanin-concentratin hormone receptor 1(MCH1-R, IC50 = 65 nM) and also inhibits hERG.
|
| T5406 |
SNAP 94847
|
487051-12-7
|
|
|
|
SNAP 94847 (SNAP-94847) is a selective and competitive MCH1 receptor (MCH1-R) antagonist (Ki: 2.2 nM). It has anxiolytic and antidepressant activity and reduces ...
|
| T8004 |
SNAP 94847 hydrochloride
|
1781934-47-1
|
100%
|
|
|
SNAP 94847 hydrochloride is a melanin-concentrating hormonereceptor1 (MCHR1) antagonist(Ki= 2.2 nM)
|
| TP1578L |
Neuropeptide EI, rat acetate
|
TP1578L
|
95.55%
|
|
|
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.
|
| TP1953L |
PG 931 acetate
|
|
98.74%
|
|
|
PG 931 acetate is a potent agonist of melanocortin 4 (MC4) receptors.
|
| T13101 |
TC-MCH 7c
|
864756-35-4
|
98.8%
|
|
|
TC-MCH 7c is an oral, selectable and blood-brain barrier penetrating MCH1R antagonist with IC50 performance of 5.6 nM against hMCH1R, and TC-MCH 7c is a phenylpy...
|
| TP1997L |
[Ala17]-MCH acetate
|
TP1997L
|
98.92%
|
|
|
[Ala17]-MCH acetate is a selective ligand for MCHR1 with a Ki of 0.16 nM and Kd of 0.37 nM(Eu3+ chelate-labeled). [Ala17]-MCH acetate shows selectivity over MCHR...
|
| TP1104L |
Melanin Concentrating Hormone, salmon acetate
|
TP1104L
|
99.41%
|
|
|
Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.
|
| TP1996 |
MCH(human, mouse, rat)
|
128315-56-0
|
99.55%
|
|
|
MCH(human, mouse, rat) is a potent endogenous agonist at melanin-concentration hormone (MCH) receptors (IC50 values are 0.3 and 1.5 nM and EC50 values are 3.9 an...
|
| T22591 |
ATC 0175 hydrochloride
|
510733-97-8
|
99.84%
|
|
|
ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective. ATC 0175 hydrochloride has affini...
|
