| T20501 |
Undecylenoyl phenylalanine
|
175357-18-3
|
98%
|
|
|
Undecylenoyl phenylalanine (Sepiwhite msh QD) is a novel depigmenting agent, which possibly acts as an alpha-melanocyte-stimulating hormone antagonist, thus inhi...
|
| T25310 |
Dersimelagon
|
1835256-48-8
|
98%
|
|
|
Dersimelagon (MT-7117) is an orally active, selective agonist for the melanocortin 1 receptor (MC1R), demonstrating EC50 values of 8.16 nM (h), 3.91 nM (cm), 1.1...
|
| TP1011L |
ACTH (1-17) acetate
|
|
98%
|
|
|
ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).
|
| TP1898 |
HS024
|
212370-59-7
|
100%
|
|
|
HS024 is a highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respec...
|
| T7813 |
α-MSH
|
581-05-5
|
100%
|
|
|
α-MSH (MSH, amide) is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase.
|
| TP1324 |
Melanotan (MT)-II
|
121062-08-6
|
100%
|
|
|
Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).
|
| TP2015L |
HS 014 acetate(207678-81-7 free base)
|
TP2015L
|
100%
|
|
|
HS 014 acetate is a potent and selective melanocortin MC4 receptor antagonist (Ki values are 3.16, 108, 54.4 and 694 nM for cloned human MC4, MC1, MC3 and MC5 re...
|
| TP1893L1 |
[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
|
TP1893L1
|
100%
|
|
|
Selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively). Displays anti-inflammato...
|
| TP1248L |
ACTH 11-24 acetate(4237-93-8 free base)
|
79190-56-0
|
100%
|
|
|
ACTH 11-24 acetate(4237-93-8 free base) (Adrenocorticotropic Hormone (11-24) acetate) is a fragment of adrenocorticotrophin, induces cortisol release. ACTH (11-2...
|
| T12882L |
Setmelanotide Acetate(920014-72-8 free base)
|
2759937-80-7
|
100%
|
|
|
Setmelanotide Acetate(920014-72-8 free base) (RM-493 Acetate) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM a...
|
| TP1578L |
Neuropeptide EI, rat acetate
|
TP1578L
|
95.55%
|
|
|
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.
|
| T7608 |
Bremelanotide Acetate
|
1607799-13-2
|
98%
|
|
|
Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .
|
| T7589 |
Afamelanotide acetate
|
1566590-77-9
|
98%
|
|
|
Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist, used to for Erythropoietic Pro...
|
| TP1952L |
PG 106 acetate
|
|
98.24%
|
|
|
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with t...
|
| TP1101 |
Nonapeptide-1 acetate salt (158563-45-2 free base)
|
TP1101
|
98.26%
|
|
|
Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) , a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antag...
|
| TP2212L |
A-MSH, amide Acetate(581-05-5 free base)
|
TP2212L
|
98.67%
|
|
|
a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities....
|
| T9596 |
AP1189 acetate
|
959850-74-9
|
98.73%
|
|
|
AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.
|
| T8485 |
THIQ
|
312637-48-2
|
98.93%
|
|
|
THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).
|
| T7627L |
Adrenocorticotropic Hormone (ACTH) (4-10) TFA
|
T7627L
|
99%
|
|
|
Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) is an agonist of potent melanocortin(MC4R) receptor .
|
| T5464 |
JNJ-10229570
|
524923-88-4
|
99.06%
|
|
|
JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland differentiat...
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