| T12241 |
Norbinaltorphimine dihydrochloride
|
113158-34-2
|
98%
|
|
|
Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.
|
| TP1832 |
Gluten Exorphin C
|
142479-62-7
|
98%
|
|
|
Gluten exorphin C is an opioid peptide derived from wheat gluten. Its IC50 values are 40 μM and 13.5 μM for μ opioid and δ opioid activities in the GPI and MVD a...
|
| T20166 |
Deltorphin
|
119975-64-3
|
98%
|
|
|
Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.
|
| TP1940L1 |
Ac-RYYRIK-NH2 acetate
|
TP1940L1
|
98%
|
|
|
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity. Ac-RYYRIK-NH2 acetate is a partial ag...
|
| TP2052L |
CTOP acetate
|
TP2052L
|
98%
|
|
|
CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.
|
| TP1941L1 |
Ac-RYYRWK-NH2 acetate
|
TP1941L1
|
98%
|
|
|
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.
|
| T77445 |
Apitegromab
|
2278276-46-1
|
98%
|
Apitegromab
|
|
Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including spinal...
|
| T14551 |
Bevenopran
|
676500-67-7
|
98%
|
|
|
Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies about the treatment of opioid-induced bowel dysfunction.
|
| T0918 |
Trimebutine
|
39133-31-8
|
98%
|
|
|
Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal pain with antimuscarinic and weak mu-opioid ag...
|
| T39284 |
EST73502 HCl
|
2307458-82-6
|
98%
|
|
|
EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.
|
| TP2485 |
Difelikefalin acetate(1024828-77-0 Free base)
|
TP2485
|
|
|
|
is a ketone and a building block.
|
| T13414 |
ZT 52656A hydrochloride
|
115730-24-0
|
|
|
|
ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.
|
| TP2036L |
DPDPE TFA (88373-73-3 free base)
|
172888-59-4
|
|
|
|
DPDPE TFA is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is ant...
|
| T0201 |
Meptazinol hydrochloride
|
59263-76-2
|
|
|
|
Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.
|
| T22850 |
ICI 204,448
|
121264-04-8
|
100%
|
|
|
ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.
|
| T7637 |
Deltorphin I
|
122752-15-2
|
100%
|
|
|
Deltorphin I is an agonist of δ-opioid receptor.
|
| T7748 |
Dermorphin TFA
|
78331-26-7
|
100%
|
|
|
Dermorphin TFA is a new class of opioids-like peptides
|
| T8557 |
N-terminally acetylated Leu-enkephalin
|
T8557
|
100%
|
|
|
Leu-enkephalin, an endogenous peptide consisting of five amino acids, functions as an agonist at opioid receptors. The N-terminally acetylated form of this compo...
|
| T7639 |
Deltorphin 2
|
122752-16-3
|
100%
|
|
|
Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.
|
| TP1905 |
BW-180C
|
63631-40-3
|
100%
|
|
|
BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.
|
