T1648 |
α-Vitamin E
|
59-02-9
|
98%
|
|
α-Vitamin E (Dexrabeprazole Sodium) is a naturally-occurring form of vitamin E, a fat-soluble vitamin with potent antioxidant properties.
|
T9256 |
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine
|
1071135-06-2
|
98%
|
|
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine is a novel 2,6-naphthyridine identified by high throughput screen (HTS) as a dual protein...
|
TN3694 |
Coniferaldehyde
|
20649-42-7
|
98%
|
|
Coniferaldehyde can significantly inhibit the growth of viability of strains of Oenococcus oeni. Coniferaldehyde exerts anti-inflammatory properties by inducing ...
|
T14072 |
A-443654
|
552325-16-3
|
98%
|
|
A-443654 is a pan-Akt inhibitor. A-443654 has equal potency against Akt1, Akt2, or Akt3 within cells (Ki=160 pM).
|
T7790 |
Bisindolylmaleimide V
|
113963-68-1
|
98%
|
|
Bisindolylmaleimide V, a bisindolylmaleimide derivative, is an inactive of a kinase inhibitor.
|
TN2326 |
(Z)-Butylidenephthalide
|
72917-31-8
|
98%
|
|
(Z)-Butylidenephthalide ((Z)-3-Butylidenephthalide) has antitumor and hypoglycemic effects, and can effectively inhibit the tumor growth of glioma and inhibit R-...
|
T1606 |
Fasudil
|
103745-39-7
|
98%
|
|
Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.
|
T6605 |
NH125
|
278603-08-0
|
98%
|
|
NH125 is a selective eEF-2 kinase inhibitor with IC50 of 60 nM, >125-fold selectivity over PKC, PKA, and CaMKII, and also a potent histidine kinase inhibitor.
|
T22831 |
Protein kinase inhibitor H-7 dihydrochloride
|
108930-17-2
|
98%
|
|
Protein kinase inhibitor H-7 dihydrochloride(H-7 dihydrochloride) is a potent protein kinase C (PKC) inhibitor. Protein kinase inhibitor H-7 dihydrochloride (100...
|
T3689 |
Ruboxistaurin hydrochloride
|
169939-93-9
|
98%
|
|
Ruboxistaurin hydrochloride (LY 333531 hydrochloride) is an Isozyme-selective inhibitor of protein kinase C (PKC); competitively and reversibly inhibits PKCβI an...
|
T13363 |
Y06137
|
2226534-49-0
|
98%
|
|
Y06137 is an effective and selective BET inhibitor with a Kd of 81 nM for BRD4(1) bromodomain. Y06137 can be used for research on the treatment of castration-res...
|
TP1888L1 |
[Ala113]-MBP (104-118) acetate
|
TP1888L1
|
98%
|
|
[Ala113]MBP(104-118) acetate is an noncompetitive peptide inhibitors of protein kinase C (PKC), with IC50s ranging from 28-62 μM.
|
T11665 |
Ionomycin calcium
|
56092-82-1
|
98%
|
|
lonomycin calcium is a potent, selective calcium ionophore and an antibiotic produced by Streptomyces conglobatus. also induces the activation of protein kinase ...
|
T4444 |
A-674563 HCl (552325-73-2(free base))
|
2070009-66-2
|
98%
|
|
A-674563 is an orally available, ATP-competitive, and reversible inhibitor of Akt (Ki: 11 nM for Akt1) [1]. It exhibits inhibitory activity against PKA and Cdk2 ...
|
TP1887L1 |
[Ala107]-MBP (104-118) acetate
|
TP1887L1
|
98%
|
|
[Ala107]-MBP (104-118) acetate ([Ala107]-MBP ) is synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor of PKC (IC50 = 46 - 14...
|
T60109 |
Protein kinase inhibitor H-7
|
84477-87-2
|
98%
|
|
Protein kinase inhibitor H-7 (5-(2-methylpiperazine-1-sulfonyl)isoquinoline) is a potent inhibitor of protein kinase C (PKC) with a Ki of 6 μM. Protein kinase in...
|
T77332 |
TV 3279
|
209394-29-6
|
98%
|
|
TV 3279 is a novel ChE-MAI inhibitor , and the neuroprotective properties depend on their ability to induce the anti-apoptotic proteins PKC, Bcl-2, Bcl-x, and SO...
|
T2S0531 |
Pinoresinol dimethyl ether
|
29106-36-3
|
98%
|
|
Pinoresinol dimethyl ether is a natural product for research related to life sciences. The catalog number is T2S0531 and the CAS number is 29106-36-3.
|
T35407 |
Ζ-Stat
|
3316-02-7
|
98%
|
|
ζ-Stat (NSC37044) is a specific and atypical PKC-ζ inhibitor, with an IC50 of 5 μM. ζ-Stat can reduce melanoma cell lines proliferation and induce apoptosis, and...
|
T14943 |
CGP60474
|
164658-13-3
|
98%
|
|
CGP60474 is an inhibitor of VEGFR-2 (IC50 = 84 nM) and an inhibitor of ATP-competitive PKC. CGP60474 is also a highly potent anti-endotoxemic agent and inhibits ...
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