| T8602 |
2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE
|
13947-21-2
|
98%
|
|
|
2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE targets the Neutrophil elastase (human).
|
| T8563 |
2-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one
|
1234707-32-4
|
98%
|
|
|
2-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one is an human neutrophil elastase inhibitor.
|
| T8362 |
Benzamidine hydrochloride
|
1670-14-0
|
98%
|
|
|
Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin (Ki of 35, 350, and 220 μM, r...
|
| T3359 |
Aprotinin
|
9087-70-1
|
98%
|
|
|
Aprotinin (Traskolan) a broad-spectrum serine protease inhibitor, inhibiting the activity of a number of different esterases and proteases, including trypsin, ch...
|
| T20992 |
MEGA-9
|
85261-19-4
|
98%
|
|
|
MEGA-9 (Nonanoyl-N-Methylglucamide) solubilizes membrane protein and can be used as a nonionic detergent.
|
| T6370 |
AEBSF hydrochloride
|
30827-99-7
|
98%
|
|
|
AEBSF hydrochloride (Pefabloc SC) is an irreversible inhibitor of serine proteases, such as chymotrypsin, kallikrein, thrombin, plasmin, and trypsin.
|
| T13257 |
Upamostat
|
590368-25-5
|
98%
|
|
|
Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) inhibitor.
|
| TP1792L |
KKI-5 acetate(97145-43-2 free base)
|
TP1792L
|
98%
|
|
|
KKI-5 acetate is a serine protease inhibitor that inhibits kallikrein and plasmin. KKI 5 may exhibit anticancer chemotherapeutic benefit and may also be used as ...
|
| T13408 |
ZK824190
|
2254001-81-3
|
98%
|
|
|
ZK824190 is an orally available and selective inhibitor of urokinase plasminogen activator (uPA) as a potential treatment for multiple sclerosis(IC50s of 237, 16...
|
| T6564 |
Leupeptin Hemisulfate
|
103476-89-7
|
98%
|
|
|
Leupeptin hemisulfate is a protease inhibitor with cell membrane-permeable, reversible, competitive, and oral activities. Leupeptin hemisulfate inhibits the acti...
|
| T8802 |
2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)-
|
80499-32-7
|
|
|
|
2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)- (Ulinastatin) ,as an urinary trypsin inhibitor (UTI), is a glycoprotein that is isolated from healthy human urine ...
|
| T3990 |
AA26-9
|
1312782-34-5
|
100%
|
|
|
AA26-9 is an effective and broad-spectrum inhibitor of serine hydrolase.
|
| T9670L |
Patamostat HCl
|
3031765-17-7
|
100%
|
|
|
Patamostat HCl is a highly potent and selective small molecule protease (protease) inhibitor that inhibits trypsin, fibrinolytic enzymes, and thrombin with IC50 ...
|
| T3442 |
UK-371804
|
256477-09-5
|
95.81%
|
|
|
UK-371804 is an effective and specific uPA inhibitor. It was selected as a candidate for further preClinicalal evaluation for the treatment of chronic dermal ulc...
|
| T3S0381 |
Chrysophanol 8-O-glucoside
|
13241-28-6
|
96.84%
|
|
|
Chrysophanol 8-O-glucoside and chrysophanol have mild cytotoxicity and anti-diabetic properties and can play metabolic roles in the insulin-stimulated glucose tr...
|
| T2392 |
Nafamostat mesylate
|
82956-11-4
|
97.36%
|
|
|
Nafamostat mesylate (FUT-175), a synthetic serine protease inhibitor, has been used for the treatment of allergic disorders such as asthma, allergic rhinitis and...
|
| T30519 |
BMS-363131
|
384829-65-6
|
97.82%
|
|
|
BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of <1.7 nM.
|
| T5597 |
ZT-12-037-01
|
2328073-61-4
|
98%
|
|
|
Zt-12-037-01 is a ATP competitive STK19 inhibitor（IC50 values of 23.96 nM and 27.94 nM for STK19 (WT) and STK19 (D89N),respectively).
|
| TN1372 |
Alpha-Amyrin
|
638-95-9
|
98.14%
|
|
|
Alpha-Amyrin (alpha-Amyrine) is an inhibitor of trypsin and chymotrypsin with antineoplastic effects. alpha-Amyrin can be used in studies about acting as a hepat...
|
| T25549 |
JCP174
|
126062-19-9
|
98.19%
|
|
|
JCP174 is a depalmitoylase inhibitor that enhances Toxoplasma host-cell invasion by targeting TgPPT1.
|
