| T9256 |
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine
|
1071135-06-2
|
98%
|
|
|
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine is a novel 2,6-naphthyridine identified by high throughput screen (HTS) as a dual protein...
|
| T5169 |
SGC-GAK-1
|
2226517-76-4
|
98%
|
|
|
SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).
|
| T1858 |
CID-797718
|
370586-05-3
|
98%
|
|
|
CID-797718 is a protein kinase D1 (PKD1) inhibitor.
|
| T73594 |
Chymotrypsin
|
9004-07-3
|
98%
|
|
|
Chymotrypsin (Chymotrypsin A) is a serine protease produced by the pancreas that cleaves protein chains on the carboxyl side of aromatic amino acids.
|
| T1954 |
SRPIN340
|
218156-96-8
|
98%
|
|
|
SRPIN340 (SRPK inhibitor), a serine/arginine-rich protein kinase (SRPK)-specific inhibitor, is potent for SRPK1 (IC50 = 0.89 uM).
|
| T2062 |
Kb NB 142-70
|
1233533-04-4
|
|
|
|
kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).
|
| T5456 |
WNK-IN-11
|
2123489-30-3
|
100%
|
|
|
WNK-IN-11 (Allosteric WNK Kinase Inhibitor) is an allosteric With-No-Lysine (WNK) kinase inhibitor,WNK1(IC50 : 4 nM)
|
| T11666 |
IPR-803
|
892243-35-5
|
95%
|
|
|
IPR-803 is an effective inhibitor of the uPAR·uPA protein-protein interaction (PPI) with anti-tumor activity. IPR-803 binds directly to uPAR with a Ki of 0.2 μM....
|
| T36680 |
SM1-71
|
2088179-99-9
|
96%
|
|
|
SM1-71 is a potent multi-targeted acrylamide-modified TAK1 inhibitor that inhibits MKNK2, MAP2K1/2/3/4/6/7, GAK, AAK1, BMP2K, MAP3K7, MAPKAPK5, GSK3A/B, MAPK1/3,...
|
| T8676 |
FOY 251
|
71079-09-9
|
97.06%
|
|
|
FOY 251 is a proteinase inhibitor, and is an anti-proteolytic active metabolite camostate.
|
| T2626 |
SBC-115076
|
489415-96-5
|
97.07%
|
|
|
SBC-115076 is a potent extracellular proprotein convertase subtilisin kexin type 9 (PCSK9) antagonist.
|
| T2392 |
Nafamostat mesylate
|
82956-11-4
|
97.36%
|
|
|
Nafamostat mesylate (FUT-175), a synthetic serine protease inhibitor, has been used for the treatment of allergic disorders such as asthma, allergic rhinitis and...
|
| T10547 |
BioE-1115
|
1268863-35-9
|
97.38%
|
|
|
BioE-1115 is a selective and potent inhibitor of serine-threonine protein kinase (PASK, IC50 = 4 nM). BioE-1115 is a potent inhibitor of CK2α (IC50 = 10 μM).
|
| T7017 |
WNK463
|
2012607-27-9
|
98%
|
|
|
WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).
|
| T1863 |
CID 2011756
|
638156-11-3
|
98.15%
|
|
|
CID 2011756 is an ATP-competitive and specific PKD1 inhibitor.
|
| T19763 |
Cetraxate hydrochloride
|
27724-96-5
|
98.23%
|
|
|
Cetraxate hydrochloride (DV10062) is an oral gastrointestinal medication. It has a cytoprotective effect.
|
| T24152 |
HTH-01-091
|
2000209-42-5
|
98.40%
|
|
|
HTH-01-091 is a potent and selective maternal embryonic leucine zipper kinase (MELK) inhibitor (IC50: 10.5 nM).HTH-01-091 inhibits PIM1/2/3, RIPK2, DYRK3, smMLCK...
|
| T77501 |
TAO Kinase inhibitor 2
|
850467-77-5
|
98.73%
|
|
|
TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.
|
| T13257 |
Upamostat
|
590368-25-5
|
98.8%
|
|
|
Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) inhibitor.
|
| T72025 |
PCSK9-IN-10
|
368434-98-4
|
98.85%
|
|
|
PCSK9-IN-10, a potent and orally active inhibitor of Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9), exhibits a half-maximal inhibitory concentration (IC5...
|
