| T33412 |
MitoPQ
|
1821370-28-8
|
98%
|
|
|
MitoPQ (MitoParaquat) is a mitochondria-targeted small molecule compound that selectively enhances mitochondrial superoxide and hydrogen peroxide levels and inhi...
|
| T2924 |
Phloretin
|
60-82-2
|
98%
|
|
|
Phloretin (NSC-407292) is a well-known inhibitor of eukaryotic urea transporters, blocks VacA-mediated urea and ion transport. Phloretin is a dihydrochalcone, a ...
|
| T11421 |
Glutaminase-IN-1
|
2247127-79-1
|
98%
|
|
|
Glutaminase-IN-1 (CB839 derivative), a novel 1,3,4-selenodiazepine renal-type glutaminase (KGA) variant inhibitor, showed antitumor activity in an aggressive H22...
|
| TN1740 |
Homoeriodictyol
|
446-71-9
|
98%
|
|
|
Homoeriodictyol, a naturally occurring, bitter-masking flavanone, as a promising agent to increase appetite and food intake. The flavanone homoeriodictyol can in...
|
| T4138 |
UCPH-101
|
1118460-77-7
|
98%
|
|
|
UCPH-101 is an inhibitor of excitatory amino acid transporter subtype 1 (EAAT1) with an IC50 of 0.66 μM.
|
| TN1132 |
Procyanidin A2
|
41743-41-3
|
98%
|
|
|
Procyanidin A2 is a potential precursor of 5-(3',4'-dihydroxyphenyl)-γ-valerolactone, exhibits antioxidant, anti-inflammary, anti-hyperglycemia, and anti-type 2 ...
|
| T11412 |
IPN60090
|
1853164-83-6
|
100%
|
|
|
IPN60090 is a novel, potent, orally bioavailable, renal-type glutaminase (GLS1)-specific inhibitor with an IC50 value of 31 nM for GLS1. IPN60090 has potential a...
|
| T4182 |
Lavendustin B
|
125697-91-8
|
95.72%
|
|
|
Lavendustin B is a Tyrosine Kinase Inhibitor and an inhibitor of HIV-1 integrase (IN) interaction with its cognate cellular cofactor, lens epithelium-derived gro...
|
| T4S1545 |
Licarin B
|
51020-87-2
|
98%
|
|
|
1.(-)-Licarin B (Licarine B) has anti-mycobacterial activity.
|
| T6791 |
BPTES
|
314045-39-1
|
98.06%
|
|
|
BPTES(IC50 of 0.16 μM) is an effective and specific GlutamiN/Ase GLS1 (KGA) inhibitor.
|
| T2755 |
Rhoifolin
|
17306-46-6
|
98.11%
|
|
|
Rhoifolin (Apigenin 7-O-neohesperidoside) is extracted from Turpinia arguya Seem dried leaves.
|
| T9558 |
KL-11743
|
1369452-53-8
|
98.12%
|
|
|
KL-11743 specifically blocks glucose metabolism, triggering an acute collapse in NADH pools and a striking accumulation of aspartate, indicating a dramatic shift...
|
| T15728 |
LDN-212320
|
894002-50-7
|
98.13%
|
|
|
LDN-212320 (OSU-0212320) is a glutamate transporter EAAT2 activator. It also enhances EAAT2 levels by > 6 fold at concentrations < 5 μM after 24 h.
|
| T78234 |
Brilliant Yellow
|
3051-11-4
|
98.26%
|
|
|
Brilliant Yellow (Direct Yellow 4) is a potent and selective VGLUT inhibitor, a dye that is photodegradable.
|
| T3782 |
Jujuboside A
|
55466-04-1
|
98.49%
|
|
|
Jujuboside A is a glycoside extracted from Semen Ziziphi Spinosae, having neurophysiological inhibitory effects, used as a potential therapeutic agent for the tr...
|
| T40413 |
SW157765
|
332063-87-3
|
98.67%
|
|
|
SW157765 is a selective glucose transporter GLUT8 (SLC2A8) inhibitor, a prodrug of many compounds, that selectively inhibits the uptake of fluorescent 2-deoxyglu...
|
| T3713 |
BAY-876
|
1799753-84-6
|
98.73%
|
|
|
BAY-876 is an orally active and selective inhibitor of glucose transporter 1 (GLUT1, IC50= 2 nM). BAY-876 exhibits >130-fold more selective for GLUT1 than GLUT2,...
|
| T22317 |
DRB18
|
2863686-81-9
|
98.74%
|
|
|
DRB18 is a highly effective pan-class inhibitor of glucose transporter proteins (GLUT). It significantly modulates energy-related metabolism in A549 cells by ind...
|
| T72054 |
SLC26A3-IN-1
|
307552-53-0
|
98.91%
|
|
|
SLC26A3-IN-1 is an inhibitor of the anion-exchange protein SLC26A3 with an IC50 value of 340 nM.SLC26A3 is a solute carrier (SLC) protein and a member of the SLC...
|
| TN1100 |
Nepodin
|
3785-24-8
|
99.12%
|
|
|
Nepodin has antimalarial, and anti-inflammatory activities, it shows significant cyclooxygenase (COX) inhibitory activity. Nepodin has an antidiabetic effect, wh...
|
